Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50017108
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177574(3-(4-(2-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177568(3-(4-(benzyloxy)phenylsulfonyl)-N-mesityl-6-methyl...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177576(3-(4-(3,5-dimethoxybenzyloxy)phenylsulfonyl)-N-mes...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177581(methyl 3-((4-(2-(mesitylamino)-6-methylpyridin-3-y...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177584(3-(4-ethylphenylsulfonyl)-N-mesityl-6-methylpyridi...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177572(3-(4-(3-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177582(3-((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfon...)
Affinity DataKi:  75nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177570(3-(4-(allyloxy)phenylsulfonyl)-N-mesityl-6-methylp...)
Affinity DataKi:  119nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177588(3-(3-(benzyloxy)phenylsulfonyl)-N-mesityl-6-methyl...)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177587(N-mesityl-6-methyl-3-tosylpyridin-2-amine | CHEMBL...)
Affinity DataKi:  145nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177575(4-((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfon...)
Affinity DataKi:  157nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177577(N-mesityl-3-(4-methoxyphenylsulfonyl)-6-methylpyri...)
Affinity DataKi:  198nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177571(N-mesityl-3-(3-methoxyphenylsulfonyl)-6-methylpyri...)
Affinity DataKi:  249nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177586(N-mesityl-6-methyl-3-(4-(pyridin-2-ylmethoxy)pheny...)
Affinity DataKi:  250nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177583(N-mesityl-6-methyl-3-(4-(trifluoromethoxy)phenylsu...)
Affinity DataKi:  268nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177589(5-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfony...)
Affinity DataKi:  395nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177573(4-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfony...)
Affinity DataKi:  635nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177567(3-(4-chlorobenzylsulfonyl)-N-mesityl-6-methylpyrid...)
Affinity DataKi:  857nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177579((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfonyl)...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177566(N-mesityl-4,6-dimethyl-3-tosylpyridin-2-amine | CH...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177580(N-mesityl-4,6-dimethyl-3-(m-tolylsulfonyl)pyridin-...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177585(N-mesityl-4,6-dimethyl-3-(o-tolylsulfonyl)pyridin-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177578(N-mesityl-6-methyl-5-tosylpyridin-2-amine | CHEMBL...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177569(N-mesityl-4,6-dimethyl-3-(phenylsulfonyl)pyridin-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed