Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50016968
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175878(4-bromobutyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175872(ethyl 2-{[(4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14bS)...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175892(Maslinicacid | 2alpha,3beta-dihydroxy-12-oleanen-2...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175871(benzyl (4aS,6aS,6bR,8aR,11R,12aR,12bR,14bS)-11-(ac...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175882(benzyl (4aS,6aS,6bR,8aR,11R,12aR,12bR,14bS)-11-hyd...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175886(benzyl (4aS,6aS,6bR,8aR,12aR,12bR,14bS)-11-hydroxy...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175890(2-(piperidin-1-yl)ethyl (4aS,6aS,6bR,8aR,10R,11R,1...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175884(2-(morpholin-4-yl)ethyl (4aS,6aS,6bR,8aR,10R,11R,1...)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175881(2-bromoethyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175887(2-(diethylamino)ethyl (4aS,6aS,6bR,8aR,10R,11R,12a...)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175891(4-(diethylamino)butyl (4aS,6aS,6bR,8aR,10R,11R,12a...)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175885(benzyl (4aS,6aS,6bR,8aR,10S,11R,12aR,12bR,14bS)-11...)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175883(1H-pyrazol-1-ylmethyl (4aS,6aS,6bR,8aR,10R,11R,12a...)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175874(benzyl (4aS,6aS,6bR,8aR,10S,11R,12aR,12bR,14bS)-10...)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175889(benzyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14bS)-11...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM10849(CHEMBL113 | 1,3,7-trimethyl-3,7-dihydropurine-2,6-...)
Affinity DataIC50: 1.14E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175870(4-(morpholin-4-yl)butyl (4aS,6aS,6bR,8aR,10R,11R,1...)
Affinity DataIC50: 1.21E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175873(3-epimaslinic acid | 3-epi-masilinic acid | 3-epi-...)
Affinity DataIC50: 1.44E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175877(2-hydroxyethyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,...)
Affinity DataIC50: 1.53E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175875(methyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14bS)-10...)
Affinity DataIC50: 3.93E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175880(benzyl (4aS,6aS,6bR,8aR,10S,11R,12aR,12bR,14bS)-11...)
Affinity DataIC50: 5.80E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175876(4-(piperidin-1-yl)butyl (4aS,6aS,6bR,8aR,10R,11R,1...)
Affinity DataIC50: 5.80E+5nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175879(2-{[(4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14bS)-10,11...)
Affinity DataIC50: 1.65E+6nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50175888(benzyl (4aS,6aS,6bR,8aR,10R,11R,12aR,12bR,14bS)-11...)
Affinity DataIC50: 1.71E+6nMAssay Description:Inhibitory activity against rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed