Compile Data Set for Download or QSAR
Report error Found 119 Enz. Inhib. hit(s) with all data for entry = 50016921
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175237(N-butyl-N-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole...)
Affinity DataIC50: 350nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175239(N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 490nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175247(N-benzyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175241(N-(4-methoxybenzyl)-3-phenyl-1H-thieno[2,3-c]pyraz...)
Affinity DataIC50: 510nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175234(N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175232((4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175246(3-methyl-4-(thiophene-2-carboxamido)-1H-thieno[2,3...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175235(4-(2-chlorobenzamido)-3-methyl-1H-thieno[2,3-c]pyr...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175250(methyl 2-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyr...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175245(1-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyrazol-4-...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175239(N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175252(3-methyl-4-(2-phenoxyacetamido)-1H-thieno[2,3-c]py...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175239(N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175243(N-benzyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175245(1-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyrazol-4-...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against Pak4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175247(N-benzyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175241(N-(4-methoxybenzyl)-3-phenyl-1H-thieno[2,3-c]pyraz...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175251(methyl 3-(phenylamino)-1H-thieno[2,3-c]pyrazole-5-...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175249(N-butyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbox...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175243(N-benzyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175250(methyl 2-(5-carbamoyl-3-methyl-1H-thieno[2,3-c]pyr...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175234(N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175247(N-benzyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175238(3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide | ...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175246(3-methyl-4-(thiophene-2-carboxamido)-1H-thieno[2,3...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175236(4-acetamido-3-methyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175237(N-butyl-N-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175232((4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175234(N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175241(N-(4-methoxybenzyl)-3-phenyl-1H-thieno[2,3-c]pyraz...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175232((4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against COTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175234(N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against COTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175238(3-methyl-1H-thieno[2,3-c]pyrazole-5-carboxamide | ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Pak4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175239(N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against COTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175240(N-cyclohexyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against COTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175243(N-benzyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175232((4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175242(N-butyl-N,3-dimethyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175234(N-phenethyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175243(N-benzyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbo...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175239(N-cyclohexyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175237(N-butyl-N-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175236(4-acetamido-3-methyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175232((4-methylpiperazin-1-yl)(3-phenyl-1H-thieno[2,3-c]...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Pak4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175242(N-butyl-N,3-dimethyl-1H-thieno[2,3-c]pyrazole-5-ca...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against COTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175249(N-butyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbox...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Pak4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175249(N-butyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-carbox...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PAK 4(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175240(N-cyclohexyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Pak4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175240(N-cyclohexyl-3-methyl-1H-thieno[2,3-c]pyrazole-5-c...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Akt1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50175237(N-butyl-N-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against Plk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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