Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50016888
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174854(N-(((1R,3S)-3-(9-chloro-3-methyl-4-oxoisoxazolo[4,...)
Affinity DataEC50:  180nMAssay Description:Inhibitory activity against MRP1 in HeLa-T5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174852(rac-N-((3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]...)
Affinity DataEC50:  250nMAssay Description:Inhibitory activity against MRP1 in HeLa-T5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174855(rac-N-((3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]...)
Affinity DataEC50:  420nMAssay Description:Inhibitory activity against MRP1 in HeLa-T5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174853(rac-N-((3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]...)
Affinity DataEC50:  640nMAssay Description:Inhibitory activity against MRP1 in HeLa-T5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174854(N-(((1R,3S)-3-(9-chloro-3-methyl-4-oxoisoxazolo[4,...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against MRP1-mediated LTC4 uptake into membrane vesicles from HeLa-T5 cells expressing MRP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174852(rac-N-((3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]...)
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against MRP1-mediated LTC4 uptake into membrane vesicles from HeLa-T5 cells expressing MRP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174853(rac-N-((3-(9-chloro-3-methyl-4-oxoisoxazolo[4,3-c]...)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibitory activity against MRP1-mediated LTC4 uptake into membrane vesicles from HeLa-T5 cells expressing MRP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed