Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50016850
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235(CHEMBL16699 | 9-Hydroxy-2,5,11-trimethyl-6H-pyrido...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 3(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(CHEMBL26559 | 5,11-Dimethyl-6H-pyrido[4,3-b]carbaz...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(CHEMBL26559 | 5,11-Dimethyl-6H-pyrido[4,3-b]carbaz...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(CHEMBL26559 | 5,11-Dimethyl-6H-pyrido[4,3-b]carbaz...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235(CHEMBL16699 | 9-Hydroxy-2,5,11-trimethyl-6H-pyrido...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 3(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235(CHEMBL16699 | 9-Hydroxy-2,5,11-trimethyl-6H-pyrido...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174412(CHEMBL19954 | cid_72512 | 9-Methoxy-5,11-dimethyl-...)
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004227(CHEMBL26559 | 5,11-Dimethyl-6H-pyrido[4,3-b]carbaz...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004235(CHEMBL16699 | 9-Hydroxy-2,5,11-trimethyl-6H-pyrido...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174412(CHEMBL19954 | cid_72512 | 9-Methoxy-5,11-dimethyl-...)
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 3(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174411(N,N-Diethyl-N'-(10-methyl-11H-pyrido[3',2':4,5]pyr...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor alpha(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174407(N,N-Diethyl-N'-(9-methoxy-5-methyl-6H-pyrido[4,3-b...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174411(N,N-Diethyl-N'-(10-methyl-11H-pyrido[3',2':4,5]pyr...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174407(N,N-Diethyl-N'-(9-methoxy-5-methyl-6H-pyrido[4,3-b...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | TCMDC-12...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | TCMDC-12...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Cnrs Umr-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed