Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50000497
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.337nMAssay Description:Inhibition of [3H]QNB binding to muscarinic acetylcholine receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453183(CHEMBL2114060)
Affinity DataKi:  0.423nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.459nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic acetylcholine receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453183(CHEMBL2114060)
Affinity DataKi:  0.522nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453188(CHEMBL2115124)
Affinity DataKi:  0.533nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453188(CHEMBL2115124)
Affinity DataKi:  0.876nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453183(CHEMBL2114060)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453182(CHEMBL2114061)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453182(CHEMBL2114061)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453188(CHEMBL2115124)
Affinity DataKi:  4.10nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453186(CHEMBL2115125)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453182(CHEMBL2114061)
Affinity DataKi:  6.10nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453186(CHEMBL2115125)
Affinity DataKi:  8.30nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic acetylcholine receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453186(CHEMBL2115125)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50229584(PILOCARBINE)
Affinity DataKi:  83nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic acetylcholine receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453184(CHEMBL2115122)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50229584(PILOCARBINE)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of [3H]QNB binding to muscarinic acetylcholine receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453189(CHEMBL2114058)
Affinity DataKi:  1.43E+3nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006546(CHEMBL67700 | Acetic acid 2-benzyl-2-aza-bicyclo[2...)
Affinity DataKi:  1.56E+3nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453187(CHEMBL2115123)
Affinity DataKi:  2.26E+3nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453187(CHEMBL2115123)
Affinity DataKi:  2.57E+3nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006549(CHEMBL304551 | Acetic acid 2-methyl-2-aza-bicyclo[...)
Affinity DataKi:  5.37E+3nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453190(CHEMBL2114059)
Affinity DataKi:  6.63E+3nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453190(CHEMBL2114059)
Affinity DataKi:  7.01E+3nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453190(CHEMBL2114059)
Affinity DataKi:  7.21E+3nMAssay Description:Inhibition of [3H]- Oxo-M binding to muscarinic receptor of rat brain membrane preparationsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453184(CHEMBL2115122)
Affinity DataKi:  9.84E+3nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453184(CHEMBL2115122)
Affinity DataKi:  1.01E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006546(CHEMBL67700 | Acetic acid 2-benzyl-2-aza-bicyclo[2...)
Affinity DataKi:  1.03E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453189(CHEMBL2114058)
Affinity DataKi:  1.15E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453184(CHEMBL2115122)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006546(CHEMBL67700 | Acetic acid 2-benzyl-2-aza-bicyclo[2...)
Affinity DataKi:  1.48E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453190(CHEMBL2114059)
Affinity DataKi:  1.51E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453187(CHEMBL2115123)
Affinity DataKi:  1.53E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453189(CHEMBL2114058)
Affinity DataKi:  1.74E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006549(CHEMBL304551 | Acetic acid 2-methyl-2-aza-bicyclo[...)
Affinity DataKi:  1.75E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453184(CHEMBL2115122)
Affinity DataKi:  1.75E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453190(CHEMBL2114059)
Affinity DataKi:  1.88E+4nMAssay Description:Inhibition of [3H]QNB binding to m3 receptor transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  1.88E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic acetylcholine receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006546(CHEMBL67700 | Acetic acid 2-benzyl-2-aza-bicyclo[2...)
Affinity DataKi:  1.89E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453187(CHEMBL2115123)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat brain membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006549(CHEMBL304551 | Acetic acid 2-methyl-2-aza-bicyclo[...)
Affinity DataKi:  2.16E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453189(CHEMBL2114058)
Affinity DataKi:  2.19E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M1 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006549(CHEMBL304551 | Acetic acid 2-methyl-2-aza-bicyclo[...)
Affinity DataKi:  2.49E+4nMAssay Description:Inhibition of [3H]QNB binding to muscarinic receptor of rat heart membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006546(CHEMBL67700 | Acetic acid 2-benzyl-2-aza-bicyclo[2...)
Affinity DataKi:  2.69E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453189(CHEMBL2114058)
Affinity DataKi:  2.77E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50006549(CHEMBL304551 | Acetic acid 2-methyl-2-aza-bicyclo[...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50453187(CHEMBL2115123)
Affinity DataKi:  4.76E+4nMAssay Description:Inhibition of [3H]QNB binding to Muscarinic acetylcholine receptor M3 transfected with CHO cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed