Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50016665
TargetIntegrase(Human immunodeficiency virus type 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171810(5-(1,3-Dimethyl-2,6-dioxo-hexahydro-pyrimidin-4-yl...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of strand transfer for HIV-1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171809(5-(2,6-Dioxo-hexahydro-pyrimidin-4-yl)-8-hydroxy-[...)
Affinity DataIC50: 11nMAssay Description:Inhibition of strand transfer for HIV-1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171812(8-Hydroxy-5-(3-methyl-2,6-dioxo-hexahydro-pyrimidi...)
Affinity DataIC50: 13nMAssay Description:Inhibition of strand transfer for HIV-1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50171811(8-Hydroxy-5-(1-methyl-2,6-dioxo-hexahydro-pyrimidi...)
Affinity DataIC50: 13nMAssay Description:Inhibition of strand transfer for HIV-1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM28236(CHEMBL199145 | N-[(4-fluorophenyl)methyl]-8-hydrox...)
Affinity DataIC50: 33nMAssay Description:Inhibition of strand transfer for HIV-1 integraseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed