Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50016660
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171744(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 8.90nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171741(3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-ylmethyl)-5H-...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171747(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171733(3-Morpholin-4-ylmethyl-5H-phenanthridin-6-one | CH...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27718(CHEMBL194482 | 2-[3-(4-Phenyl-3,6-dihydro-2H-pyrid...)
Affinity DataIC50: 46nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27716(4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]...)
Affinity DataIC50: 64nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27497(2-Dimethylamino-N-(6-oxo-5,6-dihydro-phenanthridin...)
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171739(4-(5-Morpholin-4-yl-pentyl)-2H-phthalazin-1-one | ...)
Affinity DataIC50: 119nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171737(2-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]...)
Affinity DataIC50: 119nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171748(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171738(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 249nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171731(6-Methyl-2-[3-(4-phenyl-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataIC50: 274nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171742(2-Methyl-3,4a,5,7,8,8a-hexahydro-thiopyrano[4,3-d]...)
Affinity DataIC50: 467nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171736(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 495nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171732(4-(4-Morpholin-4-yl-butyl)-2H-phthalazin-1-one | C...)
Affinity DataIC50: 950nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171735(6-Methyl-2-[3-(4-phenyl-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataIC50: 6.10E+3nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171740(2-[3-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-propyl...)
Affinity DataIC50: 8.60E+3nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50171746(6,6-Dimethyl-2-[3-(4-phenyl-3,6-dihydro-2H-pyridin...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibitory concentration against Poly(ADP-ribose) polymerase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed