Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50016648
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171539(4-(4-But-2-ynyloxy-benzenesulfonyl)-thiomorpholine...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171539(4-(4-But-2-ynyloxy-benzenesulfonyl)-thiomorpholine...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171538(4-(4-But-2-ynyloxy-benzenesulfonyl)-morpholine-3-c...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171538(4-(4-But-2-ynyloxy-benzenesulfonyl)-morpholine-3-c...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171536(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methanesulfo...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171536(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methanesulfo...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171536(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methanesulfo...)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against matrix metallopeptidase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against matrix metallopeptidase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171536(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methanesulfo...)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171534(1-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-2-c...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171534(1-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-2-c...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171540(4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxycarba...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171540(4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxycarba...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171540(4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxycarba...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171540(4-(4-But-2-ynyloxy-benzenesulfonyl)-3-hydroxycarba...)
Affinity DataIC50: 9nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171539(4-(4-But-2-ynyloxy-benzenesulfonyl)-thiomorpholine...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171543(4-(4-But-2-ynyloxy-benzenesulfonyl)-2,2-dimethyl-t...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against matrix metallopeptidase 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171539(4-(4-But-2-ynyloxy-benzenesulfonyl)-thiomorpholine...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171537(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(thiophene-2...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171537(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-(thiophene-2...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171535(4-Acetyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-piper...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171535(4-Acetyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-piper...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171534(1-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-2-c...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against matrix metallopeptidase 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171539(4-(4-But-2-ynyloxy-benzenesulfonyl)-thiomorpholine...)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against matrix metallopeptidase 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171535(4-Acetyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-piper...)
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171535(4-Acetyl-1-(4-but-2-ynyloxy-benzenesulfonyl)-piper...)
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171534(1-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-2-c...)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171534(1-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-2-c...)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against matrix metallopeptidase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against matrix metallopeptidase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171538(4-(4-But-2-ynyloxy-benzenesulfonyl)-morpholine-3-c...)
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171538(4-(4-But-2-ynyloxy-benzenesulfonyl)-morpholine-3-c...)
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171544(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pentanoyl-pi...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171542(4-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-1,3...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171542(4-(4-But-2-ynyloxy-benzenesulfonyl)-piperazine-1,3...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171545(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pyridin-3-yl...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171545(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pyridin-3-yl...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171544(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pentanoyl-pi...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50171541(9-(4-But-2-ynyloxy-benzenesulfonyl)-6-thia-9-aza-s...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against TACE[ADAM metallopeptidase domain 17] in isolated enzyme assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171545(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pyridin-3-yl...)
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171545(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-pyridin-3-yl...)
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against matrix metallopeptidase 13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171536(1-(4-But-2-ynyloxy-benzenesulfonyl)-4-methanesulfo...)
Affinity DataIC50: 51nMAssay Description:Inhibitory activity against matrix metallopeptidase 9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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