Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50016601
LigandChemical structure of BindingDB Monomer ID 50171117BDBM50171117({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171106BDBM50171106((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[3-bromo-4-...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171117BDBM50171117({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171106BDBM50171106((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[3-bromo-4-...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171096BDBM50171096({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171096BDBM50171096({4-[[3-Bromo-4-(difluoro-phosphono-methyl)-benzyl]...)
Affinity DataKi:  53nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171100BDBM50171100({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-[1,2...)
Affinity DataKi:  56nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171091BDBM50171091({4-[[4-(Difluoro-phosphono-methyl)-3-methoxy-benzy...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171100BDBM50171100({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-[1,2...)
Affinity DataIC50: 74nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171099BDBM50171099([(4-{[Benzenesulfonyl-(4-[1,2,3]thiadiazol-4-yl-be...)
Affinity DataKi:  98nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171109BDBM50171109({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-meth...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171099BDBM50171099([(4-{[Benzenesulfonyl-(4-[1,2,3]thiadiazol-4-yl-be...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171097BDBM50171097({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-[1,2...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171118BDBM50171118((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[4-(difluor...)
Affinity DataKi:  590nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171101BDBM50171101((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171118BDBM50171118((4-{[(Benzyl-methyl-carbamoyl)-methyl]-[4-(difluor...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171098BDBM50171098((4-{(4-Benzoylamino-benzyl)-[4-(difluoro-phosphono...)
Affinity DataIC50: 630nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171103BDBM50171103((4-{(3-Acetyl-benzyl)-[4-(difluoro-phosphono-methy...)
Affinity DataIC50: 770nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171094BDBM50171094((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171105BDBM50171105((4-{[4-(Difluoro-phosphono-methyl)-benzyl]-thiophe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171123BDBM50171123({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-dime...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171124BDBM50171124({4-[[4-(Difluoro-phosphono-methyl)-3-methoxy-benzy...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171112BDBM50171112(({4-[(Benzenesulfonyl-benzyl-amino)-methyl]-phenyl...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171115BDBM50171115((3-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171120BDBM50171120((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171121BDBM50171121({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(4-[1,2...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171114BDBM50171114(5-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-s...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171116BDBM50171116((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171104BDBM50171104((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171108BDBM50171108((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171093BDBM50171093((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171122BDBM50171122((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171112BDBM50171112(({4-[(Benzenesulfonyl-benzyl-amino)-methyl]-phenyl...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171095BDBM50171095((4-{Benzyl-[4-(difluoro-phosphono-methyl)-benzyl]-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171092BDBM50171092({4-[[4-(Difluoro-phosphono-methyl)-benzyl]-(2-oxo-...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171110BDBM50171110([Difluoro-(4-{[(4-hydroxy-benzoyl)-(4-[1,2,3]thiad...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171111BDBM50171111([(4-{[Benzyl-(2-nitro-benzenesulfonyl)-amino]-meth...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171107BDBM50171107((4-{(2-Acetylamino-ethyl)-[4-(difluoro-phosphono-m...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171113BDBM50171113([2-(4-{[Benzyl-(2-nitro-benzenesulfonyl)-amino]-me...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171119BDBM50171119((Difluoro-{4-[(4-[1,2,3]thiadiazol-4-yl-benzylamin...)
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50171102BDBM50171102([4-({[(Benzyl-methyl-carbamoyl)-methyl]-[4-(difluo...)
Affinity DataIC50: 6.75E+4nMAssay Description:Inhibitory activity against protein tyrosine phosphatase 1B using O-methyl fluorescein monophosphateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed