Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 5509
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  5.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  6.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  8.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  14.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  17.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86716(NSC_216215 | CAS_63540-28-3 | CHEMBL239800 | Fenob...)
Affinity DataKi:  40.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86716(NSC_216215 | CAS_63540-28-3 | CHEMBL239800 | Fenob...)
Affinity DataKi:  50.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86716(NSC_216215 | CAS_63540-28-3 | CHEMBL239800 | Fenob...)
Affinity DataKi:  53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86716(NSC_216215 | CAS_63540-28-3 | CHEMBL239800 | Fenob...)
Affinity DataKi:  56.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86716(NSC_216215 | CAS_63540-28-3 | CHEMBL239800 | Fenob...)
Affinity DataKi:  58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86715(CAS_5311432 | NSC_5311432 | SIB-1893)
Affinity DataKi:  219nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86715(CAS_5311432 | NSC_5311432 | SIB-1893)
Affinity DataKi:  243nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86717(CAS_5218788 | NSC_5218788 | CHEMBL88553 | SIB-1757)
Affinity DataKi:  328nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86715(CAS_5311432 | NSC_5311432 | SIB-1893)
Affinity DataKi:  334nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86717(CAS_5218788 | NSC_5218788 | CHEMBL88553 | SIB-1757)
Affinity DataKi:  346nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86717(CAS_5218788 | NSC_5218788 | CHEMBL88553 | SIB-1757)
Affinity DataKi:  357nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86715(CAS_5311432 | NSC_5311432 | SIB-1893)
Affinity DataKi:  423nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86717(CAS_5218788 | NSC_5218788 | CHEMBL88553 | SIB-1757)
Affinity DataKi:  486nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86715(CAS_5311432 | NSC_5311432 | SIB-1893)
Affinity DataKi:  800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86717(CAS_5218788 | NSC_5218788 | CHEMBL88553 | SIB-1757)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86211(NSC_40539 | CAS_52809-07-1 | Quisqualate)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86211(NSC_40539 | CAS_52809-07-1 | Quisqualate)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86211(NSC_40539 | CAS_52809-07-1 | Quisqualate)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM86211(NSC_40539 | CAS_52809-07-1 | Quisqualate)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50002371(Glutaminsaeure | glutamic acid | Glutamate | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50002371(Glutaminsaeure | glutamic acid | Glutamate | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50002371(Glutaminsaeure | glutamic acid | Glutamate | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
F. Hoffmann-La Roche

Curated by PDSP Ki Database
LigandPNGBDBM50002371(Glutaminsaeure | glutamic acid | Glutamate | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2012
Entry Details Article
PubMed