Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50016477
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169540(Cyclopropylmethyl-(2,2,2-trifluoro-ethyl)-[2-trifl...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169535(Dipropyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-phe...)
Affinity DataKi:  11nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169517(Cyclopropylmethyl-[2-trifluoromethyl-9-(2,4,6-trim...)
Affinity DataKi:  13nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169508(Cyclopropylmethyl-[2-methyl-9-(2,4,6-trimethyl-phe...)
Affinity DataKi:  20nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169531(Cyclopropylmethyl-[2-ethyl-9-(2,4,6-trimethyl-phen...)
Affinity DataKi:  21nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169524(Cyclopropylmethyl-propyl-[2-trifluoromethyl-9-(2,4...)
Affinity DataKi:  23nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169520(Cyclobutylmethyl-propyl-[2-trifluoromethyl-9-(2,4,...)
Affinity DataKi:  26nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169533(Cyclopropylmethyl-ethyl-[2-trifluoromethyl-9-(2,4,...)
Affinity DataKi:  28nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169523(Cyclopropylmethyl-(2,2,3,3,3-pentafluoro-propyl)-[...)
Affinity DataKi:  34nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169498(Cyclobutylmethyl-(2,2,2-trifluoro-ethyl)-[2-triflu...)
Affinity DataKi:  53nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169537([9-(2-Bromo-4-isopropyl-phenyl)-2-trifluoromethyl-...)
Affinity DataKi:  54nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169529(Cyclopropylmethyl-[6-fluoro-2-methyl-9-(2,4,6-trim...)
Affinity DataKi:  59nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169526(Propyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-pheny...)
Affinity DataKi:  68nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169515(Propyl-(2,2,2-trifluoro-ethyl)-[2-trifluoromethyl-...)
Affinity DataKi:  75nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169511((2,2,3,3,3-Pentafluoro-propyl)-propyl-[2-trifluoro...)
Affinity DataKi:  75nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169507(Diallyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-phen...)
Affinity DataKi:  138nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169509(Cyclopropylmethyl-[2-ethyl-6-fluoro-9-(2,4,6-trime...)
Affinity DataKi:  150nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169505([9-(2-Bromo-4-isopropyl-phenyl)-2-trifluoromethyl-...)
Affinity DataKi:  150nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169539(Bis-cyclopropylmethyl-[9-(2,4-dichloro-phenyl)-2-t...)
Affinity DataKi:  240nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169534(Ethyl-phenethyl-[2-trifluoromethyl-9-(2,4,6-trimet...)
Affinity DataKi:  249nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169534(Ethyl-phenethyl-[2-trifluoromethyl-9-(2,4,6-trimet...)
Affinity DataKi:  249nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169522(Phenethyl-propyl-[2-trifluoromethyl-9-(2,4,6-trime...)
Affinity DataKi:  250nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169518((2,2,2-Trifluoro-ethyl)-[2-trifluoromethyl-9-(2,4,...)
Affinity DataKi:  291nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169512(Diphenethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-...)
Affinity DataKi:  333nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169519(2-Methyl-9-(2,4,6-trimethyl-phenyl)-9H-benzo[d]imi...)
Affinity DataKi:  360nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169501((2-Cyclopropyl-ethyl)-propyl-[2-trifluoromethyl-9-...)
Affinity DataKi:  362nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169510(Cyclopropylmethyl-[9-(2,4-dichloro-phenyl)-2-trifl...)
Affinity DataKi:  370nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169536([9-(2-Bromo-4-isopropyl-phenyl)-2-trifluoromethyl-...)
Affinity DataKi:  410nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169506(Benzyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-pheny...)
Affinity DataKi:  428nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169504((2-Cyclopropyl-ethyl)-[2-trifluoromethyl-9-(2,4,6-...)
Affinity DataKi:  457nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169527(2-Ethyl-9-(2,4,6-trimethyl-phenyl)-9H-benzo[d]imid...)
Affinity DataKi:  570nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169499(Benzyl-methyl-[2-trifluoromethyl-9-(2,4,6-trimethy...)
Affinity DataKi:  573nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169516(Phenethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-ph...)
Affinity DataKi:  618nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169502((2-Cyclopropyl-ethyl)-(2,2,2-trifluoro-ethyl)-[2-t...)
Affinity DataKi:  653nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169500(Butyl-ethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl-...)
Affinity DataKi:  704nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169525(Phenethyl-(2,2,2-trifluoro-ethyl)-[2-trifluorometh...)
Affinity DataKi:  744nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169514(2-Ethyl-6-fluoro-9-(2,4,6-trimethyl-phenyl)-9H-ben...)
Affinity DataKi:  930nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169530(6-Fluoro-2-methyl-9-(2,4,6-trimethyl-phenyl)-9H-be...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169538((2-Cyclopropyl-ethyl)-ethyl-[2-trifluoromethyl-9-(...)
Affinity DataKi:  1.41E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169528([9-(2,4-Dichloro-phenyl)-2-trifluoromethyl-9H-benz...)
Affinity DataKi:  1.60E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169503(Benzyl-ethyl-[2-trifluoromethyl-9-(2,4,6-trimethyl...)
Affinity DataKi:  2.77E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169532(2-Trifluoromethyl-9-(2,4,6-trimethyl-phenyl)-9H-be...)
Affinity DataKi:  3.56E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169513(Benzyl-propyl-[2-trifluoromethyl-9-(2,4,6-trimethy...)
Affinity DataKi:  4.05E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50169521(Benzyl-butyl-[2-trifluoromethyl-9-(2,4,6-trimethyl...)
Affinity DataKi:  7.71E+3nMAssay Description:Binding affinity for human corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed