Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50016374
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168291(Sodium; {3-[(S)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi:  54nMAssay Description:Inhibition of [3H]-Iloprost binding to human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  930nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Prostanoid TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]SQ-29,548 binding to human Prostanoid TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-PGF-2 binding to human Prostanoid FP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]PGD-2 binding to human Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi:  1.02E+3nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of [3H]PGD-2 binding to human Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136234(Sodium; {3-[(R)-2-(4,5-diphenyl-oxazol-2-yl)-cyclo...)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of [3H]-PGE-2 binding to Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi:  7.20E+3nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]-PGF-2 binding to human Prostanoid FP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50168287(Sodium; {3-[(1R,2S,6S)-1-(4,5-diphenyl-oxazol-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]PGE-2 binding to Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed