Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50003697
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474925(CHEMBL294757)
Affinity DataKi:  1.80nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50004108((R,S)-nicotine | (RS)-nicotine | nicotine | (+-)-n...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474921(CHEMBL103225)
Affinity DataKi:  5.60nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474922(CHEMBL190652)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474928(CHEMBL103537)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474927(CHEMBL191253)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50004108((R,S)-nicotine | (RS)-nicotine | nicotine | (+-)-n...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]epibatidine binding to rat Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474924(CHEMBL189470)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474923(CHEMBL361703)
Affinity DataKi:  72nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  200nMAssay Description:Inhibition of [3H]epibatidine binding to rat Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474926(CHEMBL363379)
Affinity DataKi:  275nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474929(CHEMBL190678)
Affinity DataKi:  350nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  400nMAssay Description:Binding affinity for rat Nicotinic acetylcholine receptor alpha4-beta4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  490nMAssay Description:Binding affinity for rat Nicotinic acetylcholine receptor alpha2-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity for rat Nicotinic acetylcholine receptor alpha2-beta4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity for rat Nicotinic acetylcholine receptor alpha3-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50168255((+/-)6-(2-Phenylethyl)nicotine | 5-(1-Methyl-pyrro...)
Affinity DataKi:  4.60E+3nMAssay Description:Binding affinity for rat Nicotinic acetylcholine receptor alpha3-beta4More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50451799(CHEMBL350748)
Affinity DataKi:  9.44E+3nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474920(CHEMBL190618)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474930(CHEMBL370709)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50474923(CHEMBL361703)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H](-)-nicotine binding to rat brain (minus cerebellum) Nicotinic acetylcholine receptor alpha4-beta2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed