Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50037396
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892({(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydro...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891({6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahy...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]iloprost from human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892({(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGD-2 from human Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SQ-29,548 from human Prostanoid TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGF-2 from human Prostanoid FP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892({(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydro...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]SQ-29,548 from human Prostanoid TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891({6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGD-2 from human Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891({6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PGF-2 from human Prostanoid FP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891({6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahy...)
Affinity DataKi: >1.90E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin D2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]PGD-2 from human Prostanoid DP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50370452(FR-181157 | CHEMBL132589)
Affinity DataKi:  6.80E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi:  8.20E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi:  9.60E+3nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892({(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SQ-29,548 from human Prostanoid TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP2 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-PGE-2 from human Prostanoid EP2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167891({6-[(Diphenylcarbamoyloxy)-methyl]-5,6,7,8-tetrahy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin F2-alpha receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167887({(R)-6-[(Diphenylcarbamoyloxy)-methyl]-6-hydroxy-5...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGF-2 from human Prostanoid FP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167890(FR-193262 | Sodium; {(R)-5-[(R)-2-(4,5-diphenyl-ox...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50167892({(S)-6-[(Diphenylcarbamoyloxy)-methyl]-5,6-dihydro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PGE-2 from human Prostanoid EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed