Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50037394
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167871(3-Chloro-4-{4-[5-(4-methyl-pyrimidin-2-yl)-3,4-dih...)
Affinity DataIC50: 0.185nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50097341(3-Chloro-4-[4-(4-pyridin-2-yl-piperazin-1-yl)-buty...)
Affinity DataIC50: 0.770nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167872(3-Chloro-4-[4-(4-pyrimidin-2-yl-3,6-dihydro-2H-pyr...)
Affinity DataIC50: 1.38nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50097343(3-Chloro-4-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-bu...)
Affinity DataIC50: 1.59nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167869(3-Chloro-4-[4-(4-pyrimidin-2-yl-piperidin-1-yl)-bu...)
Affinity DataIC50: 5.81nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50097341(3-Chloro-4-[4-(4-pyridin-2-yl-piperazin-1-yl)-buty...)
Affinity DataIC50: 51nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167870(3-Chloro-4-[4-(5-pyrimidin-2-yl-3,6-dihydro-2H-pyr...)
Affinity DataIC50: 79.6nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50097343(3-Chloro-4-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-bu...)
Affinity DataIC50: 199nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167874(3-Chloro-4-[4-(3-pyrimidin-2-yl-piperidin-1-yl)-bu...)
Affinity DataIC50: 324nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167872(3-Chloro-4-[4-(4-pyrimidin-2-yl-3,6-dihydro-2H-pyr...)
Affinity DataIC50: 494nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167871(3-Chloro-4-{4-[5-(4-methyl-pyrimidin-2-yl)-3,4-dih...)
Affinity DataIC50: 763nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167870(3-Chloro-4-[4-(5-pyrimidin-2-yl-3,6-dihydro-2H-pyr...)
Affinity DataIC50: 893nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167869(3-Chloro-4-[4-(4-pyrimidin-2-yl-piperidin-1-yl)-bu...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against Dopamine receptor D2 in rat striatum membrane using [3H]raclopride as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Daiichi Suntory Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50167873(3-Chloro-4-[4-(4-hydroxy-4-pyrimidin-2-yl-piperidi...)
Affinity DataIC50: 2.65E+3nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed