Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50037499
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157335(CHEMBL1182177 | CHEMBL540872 | CHEMBL216829 | 4-(2...)
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157342(7-(3,4,5,6-Tetrahydro-2H-[1,4']bipyridinyl-4-ylmet...)
Affinity DataIC50: 56nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157330(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 74nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157339(CHEMBL195428 | CHEMBL534707 | 4-(2-Carbamimidoyl-1...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157334(3-[4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157332(3-[4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 190nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157343(CHEMBL537188 | 4-(2-Carbamimidoyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167018(4-[2-(2-Carbamimidoyl-1,2,3,4,4a,8a-hexahydro-isoq...)
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157338(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 270nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167017(4-(7-Carbamimidoyl-naphthalen-2-ylsulfanylmethyl)-...)
Affinity DataIC50: 390nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167023(1-(4-Carbamimidoyl-phenyl)-4-(2-carbamimidoyl-1,2,...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157328(7-(1-Quinolin-4-yl-piperidin-4-ylmethoxy)-3,4-dihy...)
Affinity DataIC50: 420nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157327(7-[1-(1-Imino-ethyl)-piperidin-4-ylmethoxy]-3,4-di...)
Affinity DataIC50: 510nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167020(4-(7-Carbamimidoyl-naphthalen-2-yloxymethyl)-3,4,5...)
Affinity DataIC50: 510nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157340(7-(1-Pyridin-4-ylmethyl-piperidin-4-ylmethoxy)-3,4...)
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167027(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157345(7-(1-Pyridin-2-ylmethyl-piperidin-4-ylmethoxy)-3,4...)
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157331(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167019(4-(7-Carbamimidoyl-naphthalene-2-sulfonylamino)-3,...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167028(7-[1-(2-Amino-benzyl)-piperidin-4-ylmethoxy]-3,4-d...)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157329(7-(Piperidin-4-ylmethoxy)-3,4-dihydro-1H-isoquinol...)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167021(7-[1-(3-Amino-benzyl)-piperidin-4-ylmethoxy]-3,4-d...)
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167026(7-(1-Acetyl-piperidin-4-ylmethoxy)-3,4-dihydro-1H-...)
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167024(4-(7-Carbamimidoyl-naphthalene-2-sulfonylmethyl)-3...)
Affinity DataIC50: 5.44E+3nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157340(7-(1-Pyridin-4-ylmethyl-piperidin-4-ylmethoxy)-3,4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157339(CHEMBL195428 | CHEMBL534707 | 4-(2-Carbamimidoyl-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157327(7-[1-(1-Imino-ethyl)-piperidin-4-ylmethoxy]-3,4-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157329(7-(Piperidin-4-ylmethoxy)-3,4-dihydro-1H-isoquinol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167030(4-(2-Carbamimidoyl-2,3,4,5-tetrahydro-1H-benzo[c]a...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor XMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157328(7-(1-Quinolin-4-yl-piperidin-4-ylmethoxy)-3,4-dihy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167030(4-(2-Carbamimidoyl-2,3,4,5-tetrahydro-1H-benzo[c]a...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157338(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167020(4-(7-Carbamimidoyl-naphthalen-2-yloxymethyl)-3,4,5...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167024(4-(7-Carbamimidoyl-naphthalene-2-sulfonylmethyl)-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167018(4-[2-(2-Carbamimidoyl-1,2,3,4,4a,8a-hexahydro-isoq...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167017(4-(7-Carbamimidoyl-naphthalen-2-ylsulfanylmethyl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167019(4-(7-Carbamimidoyl-naphthalene-2-sulfonylamino)-3,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167021(7-[1-(3-Amino-benzyl)-piperidin-4-ylmethoxy]-3,4-d...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157335(CHEMBL1182177 | CHEMBL540872 | CHEMBL216829 | 4-(2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167023(1-(4-Carbamimidoyl-phenyl)-4-(2-carbamimidoyl-1,2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157334(3-[4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157331(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157343(CHEMBL537188 | 4-(2-Carbamimidoyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167026(7-(1-Acetyl-piperidin-4-ylmethoxy)-3,4-dihydro-1H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157332(3-[4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinol...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167027(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157342(7-(3,4,5,6-Tetrahydro-2H-[1,4']bipyridinyl-4-ylmet...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50167028(7-[1-(2-Amino-benzyl)-piperidin-4-ylmethoxy]-3,4-d...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157345(7-(1-Pyridin-2-ylmethyl-piperidin-4-ylmethoxy)-3,4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetProthrombin(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50157330(4-(2-Carbamimidoyl-1,2,3,4-tetrahydro-isoquinolin-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against human Coagulation factor II (thrombin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
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