Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50016208
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataKi:  0.730nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50059841(CHEMBL278789 | (S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50060070(CHEMBL317264 | (S)-2-Amino-N-{1-[(S)-1-((R)-1-carb...)
Affinity DataKi:  5.10nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166347((S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-...)
Affinity DataKi:  10.4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166345(6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi:  57.8nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166346((S)-1-((S)-6-Hydroxy-1,2,3,4-tetrahydro-isoquinoli...)
Affinity DataKi:  216nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166342(6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi:  253nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50059841(CHEMBL278789 | (S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-...)
Affinity DataKi:  295nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166343((S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-...)
Affinity DataKi:  304nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166344(7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi:  1.62E+3nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50060070(CHEMBL317264 | (S)-2-Amino-N-{1-[(S)-1-((R)-1-carb...)
Affinity DataKi:  1.82E+3nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166342(6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166346((S)-1-((S)-6-Hydroxy-1,2,3,4-tetrahydro-isoquinoli...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166347((S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166345(6-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166344(7-Hydroxy-1,2,3,4-tetrahydro-isoquinoline-3-carbox...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50166343((S)-N-{(S)-1-[(S)-1-(Carbamoylmethyl-carbamoyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed