Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50016205
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166319(4-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 0.130nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166318((S)-1-[(2S,4S)-4-(3-Chloro-4-cyano-phenylamino)-py...)
Affinity DataIC50: 0.130nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166318((S)-1-[(2S,4S)-4-(3-Chloro-4-cyano-phenylamino)-py...)
Affinity DataIC50: 0.150nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166308((S)-1-[(2S,4S)-4-(4-Nitro-phenylamino)-pyrrolidine...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166319(4-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166308((S)-1-[(2S,4S)-4-(4-Nitro-phenylamino)-pyrrolidine...)
Affinity DataIC50: 0.180nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166320((S)-1-[(2S,4S)-4-(4-Cyano-phenylamino)-pyrrolidine...)
Affinity DataIC50: 0.190nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166309((S)-1-[(2S,4S)-4-(3,4-Dimethoxy-phenylamino)-pyrro...)
Affinity DataIC50: 0.240nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166315(6-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 0.25nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166320((S)-1-[(2S,4S)-4-(4-Cyano-phenylamino)-pyrrolidine...)
Affinity DataIC50: 0.260nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166315(6-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 0.270nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166317((S)-1-[(2S,4S)-4-(4-Methoxy-phenylamino)-pyrrolidi...)
Affinity DataIC50: 0.280nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166309((S)-1-[(2S,4S)-4-(3,4-Dimethoxy-phenylamino)-pyrro...)
Affinity DataIC50: 0.280nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166317((S)-1-[(2S,4S)-4-(4-Methoxy-phenylamino)-pyrrolidi...)
Affinity DataIC50: 0.330nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166311((S)-1-((2S,4S)-4-Phenylamino-pyrrolidine-2-carbony...)
Affinity DataIC50: 0.530nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166311((S)-1-((2S,4S)-4-Phenylamino-pyrrolidine-2-carbony...)
Affinity DataIC50: 0.530nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166312(1-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166306((S)-1-((2S,4S)-4-Phenethylamino-pyrrolidine-2-carb...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166312(1-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166306((S)-1-((2S,4S)-4-Phenethylamino-pyrrolidine-2-carb...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11113(NVP-DPP728 | cyanopyrrolidine derivative 2 | CHEMB...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11056(CHEMBL381626 | (2S)-1-[(2S)-pyrrolidin-2-ylcarbony...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM11056(CHEMBL381626 | (2S)-1-[(2S)-pyrrolidin-2-ylcarbony...)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166310((S)-1-((2S,4S)-4-Cyclohexylamino-pyrrolidine-2-car...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166321((S)-1-((2S,4S)-4-Benzylamino-pyrrolidine-2-carbony...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166310((S)-1-((2S,4S)-4-Cyclohexylamino-pyrrolidine-2-car...)
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166307(N-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 3.80nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166313(N-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166321((S)-1-((2S,4S)-4-Benzylamino-pyrrolidine-2-carbony...)
Affinity DataIC50: 4.60nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166307(N-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 5.5nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166314(6-((3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)py...)
Affinity DataIC50: 6.60nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166314(6-((3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)py...)
Affinity DataIC50: 6.70nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166313(N-[(3S,5S)-5-((S)-2-Cyano-pyrrolidine-1-carbonyl)-...)
Affinity DataIC50: 6.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Rat)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166316((S)-1-((2S,4S)-4-Amino-pyrrolidine-2-carbonyl)-pyr...)
Affinity DataIC50: 9.10nMAssay Description:Inhibitory concentration against rat dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50166316((S)-1-((2S,4S)-4-Amino-pyrrolidine-2-carbonyl)-pyr...)
Affinity DataIC50: 9.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed