Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50024631
TargetMuscarinic acetylcholine receptor M3(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50259847(cremastrine | CHEMBL480464)
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M3 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M4(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50259847(cremastrine | CHEMBL480464)
Affinity DataIC50: 498nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M4 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50259847(cremastrine | CHEMBL480464)
Affinity DataIC50: 505nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M1 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50259847(cremastrine | CHEMBL480464)
Affinity DataIC50: 1.22E+3nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M5 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50259847(cremastrine | CHEMBL480464)
Affinity DataIC50: 5.52E+3nMAssay Description:Displacement of [3H]NMS from human cloned muscarinic M2 receptor expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed