Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50016144
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50: 400nMAssay Description:Mean inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 790nMAssay Description:Mean inhibitory concentration against potassium channel HERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50: 1.32E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 3.16E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50: 5.29E+3nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50: 1.05E+4nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2B expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50: 2.49E+4nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165457((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-1,2,3...)
Affinity DataIC50: 1.04E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 1.07E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165461((S)-1-(4-Chloro-phenyl)-2-((S)-6,7-dimethoxy-2-met...)
Affinity DataIC50: 1.37E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2A expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(Rat)
Ludwig-Maximilians-UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50165458((S)-2-((S)-6,7-Dimethoxy-2-methyl-1,2,3,4-tetrahyd...)
Affinity DataIC50: 1.55E+5nMAssay Description:Mean inhibitory concentration against rat N-methyl-D-aspartate (NMDA) glutamate receptor 1a/2C expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed