Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 947
LigandPNGBDBM7440(2,4,6-Trimethyl-N-(3-oxo-1,2,3,6-tetrahydro-2,4,6-...)
Affinity DataIC50: 1.50E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7435(8-(aminomethyl)-4,7,10-triazatetracyclo[7.7.0.0^{2...)
Affinity DataIC50: 5.50E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7438(10-[2-(dimethylamino)ethyl]-8-methyl-4,7,10-triaza...)
Affinity DataIC50: 7.00E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7439(2-(dimethylamino)-N-({5-oxo-4,7,10-triazatetracycl...)
Affinity DataIC50: 8.00E+3nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7450({[({2-benzyl-4-methyl-1,3-dioxo-1H,2H,3H,5H-pyrrol...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7430(5-Methyl-6-(2-trimethylsilanyl-ethoxymethyl)-1,2-d...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7449({[({2,4-dimethyl-1,3-dioxo-1H,2H,3H,5H-pyrrolo[3,4...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7448(N-[(2-benzyl-4-methyl-1,3-dioxo-5-{[2-(trimethylsi...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7447(N-[(2,4-dimethyl-1,3-dioxo-5-{[2-(trimethylsilyl)e...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7446(N-[(2-benzyl-4-methyl-1,3-dioxo-5-{[2-(trimethylsi...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7445(N-[(2,4-dimethyl-1,3-dioxo-5-{[2-(trimethylsilyl)e...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7444(10-(aminomethyl)-2-benzyl-4-methyl-5-{[2-(trimethy...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7443(10-(aminomethyl)-2,4-dimethyl-5-{[2-(trimethylsily...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7442(2,4-dimethyl-1,3-dioxo-5-{[2-(trimethylsilyl)ethox...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7441(8-chloro-2,4-dimethyl-1,3-dioxo-5-{[2-(trimethylsi...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7437(2-(2-Dimethylaminoethyl)-5-methyl-1,2-di-hydro-6H-...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7436(5-Methyl-1,2-dihydro-6H-2,4,6-triaza-cyclopenta[c]...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7434(2-Benzyl-5-phenyl-1,2-dihydro-6H-2,4,6-triazacyclo...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7433(2-[2-(dimethylamino)ethyl]-5-methyl-6-{[2-(trimeth...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7432(4-[2-(dimethylamino)ethyl]-3-imino-8-methyl-10-{[2...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed
LigandPNGBDBM7431(8-methyl-4,10-diazatetracyclo[7.7.0.0^{2,6}.0^{11,...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/ [gamma-32P] ATP. 32...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2006
Entry Details Article
PubMed