Compile Data Set for Download or QSAR
Report error Found 137 Enz. Inhib. hit(s) with all data for entry = 50041392
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061349([2-(3-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  0.309nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061345([2-(3,4-Dimethyl-phenoxy)-ethyl]-(3-phenoxy-propyl...)
Affinity DataKi:  0.347nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061351((3-Phenoxy-propyl)-(2-m-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  0.457nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061332((3-Phenoxy-propyl)-(2-p-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061339([2-(4-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061334([2-(3-Chloro-4-methyl-phenoxy)-ethyl]-(3-phenoxy-p...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061330([2-(4-Chloro-phenoxy)-ethyl]-[3-(4-fluoro-phenoxy)...)
Affinity DataKi:  0.832nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061325([3-(4-Fluoro-phenoxy)-propyl]-(2-p-tolyloxy-ethyl)...)
Affinity DataKi:  0.955nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061324((2-p-Tolyloxy-ethyl)-(3-o-tolyloxy-propyl)-amine |...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058234(N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-4-meth...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061327((2-p-Tolyloxy-ethyl)-(3-m-tolyloxy-propyl)-amine |...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061346((2-Phenoxy-ethyl)-(3-phenoxy-propyl)-amine | CHEMB...)
Affinity DataKi:  2nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061337((2-Phenoxy-ethyl)-(3-p-tolyloxy-propyl)-amine | CH...)
Affinity DataKi:  2.69nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061336(4-[2-(3-Phenoxy-propylamino)-ethoxy]-phenol | CHEM...)
Affinity DataKi:  3.09nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058222(N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-4-me...)
Affinity DataKi:  3.39nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058223(4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  3.47nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061334([2-(3-Chloro-4-methyl-phenoxy)-ethyl]-(3-phenoxy-p...)
Affinity DataKi:  3.89nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058233(4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  3.89nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061348([2-(4-Nitro-phenoxy)-ethyl]-(3-phenoxy-propyl)-ami...)
Affinity DataKi:  4.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061340([2-(2-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  4.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50175151(3-(3-(bis(4-fluorophenyl)methoxy)-8-aza-bicyclo[3....)
Affinity DataKi:  5.01nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058230(4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  5.25nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058226(3-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  5.25nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061343([2-(4-Methoxy-phenoxy)-ethyl]-(3-phenoxy-propyl)-a...)
Affinity DataKi:  5.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058233(4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061326([2-(4-Chloro-phenoxy)-ethyl]-(3-p-tolyloxy-propyl)...)
Affinity DataKi:  5.62nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058234(N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-4-meth...)
Affinity DataKi:  6.46nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148744(N-(2-{3-[Bis-(4-fluoro-phenyl)-methoxy]-8-aza-bicy...)
Affinity DataKi:  6.46nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058232(N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-3-me...)
Affinity DataKi:  6.76nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058222(N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-4-me...)
Affinity DataKi:  7.76nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148741(Benzyl-(2-{3-[bis-(4-fluoro-phenyl)-methoxy]-8-aza...)
Affinity DataKi:  8.13nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058230(4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  8.32nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058225(N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-3-meth...)
Affinity DataKi:  8.71nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061344((2-p-Tolyloxy-ethyl)-(3-p-tolyloxy-propyl)-amine |...)
Affinity DataKi:  11.0nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058220(N-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-4-met...)
Affinity DataKi:  12.0nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058232(N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-3-me...)
Affinity DataKi:  12.9nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM86701(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-azoni...)
Affinity DataKi:  13.8nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148736(N-(2-{3-[Bis-(4-fluoro-phenyl)-methoxy]-8-aza-bicy...)
Affinity DataKi:  14.1nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058223(4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  14.1nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058228(3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  15.1nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058228(3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  15.1nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058224(N-[4-(2-Chloro-phenyl)-piperazin-1-ylmethyl]-3-met...)
Affinity DataKi:  15.8nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058225(N-[4-(2-Cyano-phenyl)-piperazin-1-ylmethyl]-3-meth...)
Affinity DataKi:  17.0nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061340([2-(2-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  17.0nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148742(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-[2-(thiophen-2...)
Affinity DataKi:  18.6nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061335((3-Phenoxy-propyl)-(2-o-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  19.9nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058231(N-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-benz...)
Affinity DataKi:  21.9nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061349([2-(3-Chloro-phenoxy)-ethyl]-(3-phenoxy-propyl)-am...)
Affinity DataKi:  21.9nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148740(8-(2-Benzyloxy-ethyl)-3-[bis-(4-fluoro-phenyl)-met...)
Affinity DataKi:  22.4nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Pomona College

Curated by ChEMBL
LigandPNGBDBM50039177(CHEMBL119664 | CHEMBL541825 | 3-[Bis-(4-chloro-phe...)
Affinity DataKi:  23.4nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
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