Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 850
LigandPNGBDBM6671(3-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 160nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 180nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 200nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6672(N-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 250nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6671(3-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 250nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6670(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 390nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6673(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 450nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6662(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-methanesulfo...)
Affinity DataIC50: 520nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6670(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 560nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM6666(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 580nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6672(N-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 670nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6673(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 740nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 960nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6668(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 970nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6662(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-methanesulfo...)
Affinity DataIC50: 1.21E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6662(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-methanesulfo...)
Affinity DataIC50: 1.22E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6671(3-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 1.29E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6670(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.34E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6668(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.54E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6666(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.61E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6666(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.63E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6663(6-[(2,6-dichlorophenyl)carbonyl]-N-(3-methanesulfo...)
Affinity DataIC50: 1.70E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6667(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.92E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6668(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 2.16E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6667(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 2.72E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6663(6-[(2,6-dichlorophenyl)carbonyl]-N-(3-methanesulfo...)
Affinity DataIC50: 2.86E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6664(6-[(2,6-dichlorophenyl)carbonyl]-N-[4-(methylsulfa...)
Affinity DataIC50: 3.04E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6663(6-[(2,6-dichlorophenyl)carbonyl]-N-(3-methanesulfo...)
Affinity DataIC50: 3.14E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6672(N-{[4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,...)
Affinity DataIC50: 3.84E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6667(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 3.95E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6665(6-[(2,6-dichlorophenyl)carbonyl]-N-[3-(methylsulfa...)
Affinity DataIC50: 4.80E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6673(4-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 4.99E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6664(6-[(2,6-dichlorophenyl)carbonyl]-N-[4-(methylsulfa...)
Affinity DataIC50: 7.40E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6669(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 9.26E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6665(6-[(2,6-dichlorophenyl)carbonyl]-N-[3-(methylsulfa...)
Affinity DataIC50: 1.19E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6669(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 1.21E+4nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6664(6-[(2,6-dichlorophenyl)carbonyl]-N-[4-(methylsulfa...)
Affinity DataIC50: 1.39E+4nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6665(6-[(2,6-dichlorophenyl)carbonyl]-N-[3-(methylsulfa...)
Affinity DataIC50: 1.77E+4nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6669(3-({6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6674(N-{6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]p...)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6675(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-phenoxypheny...)
Affinity DataIC50: 2.00E+4nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6675(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-phenoxypheny...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6674(N-{6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]p...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6675(6-[(2,6-dichlorophenyl)carbonyl]-N-(4-phenoxypheny...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed
LigandPNGBDBM6674(N-{6-[(2,6-dichlorophenyl)carbonyl]imidazo[1,2-a]p...)
Affinity DataIC50: 2.00E+4nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2005
Entry Details Article
PubMed