Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50037435
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292221((S)-3-(2,4-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50366689(GHRELIN)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292225((S)-3-(2,5-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292228((S)-3-(2,3-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50151162((S)-3-(2-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 4nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292230((S)-3-(2,6-Dichloro-phenyl)-1-(2-diethylamino-ethy...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292223((R)-3-(3-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 15nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292227((R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(3-methox...)
Affinity DataIC50: 77nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292226((R)-3-(4-Chloro-phenyl)-1-(2-diethylamino-ethyl)-3...)
Affinity DataIC50: 83nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292229((R)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(4-methox...)
Affinity DataIC50: 106nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292224(1-(2-Diethylamino-ethyl)-3-hydroxy-2-oxo-3-phenyl-...)
Affinity DataIC50: 116nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sumitomo Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292222((S)-1-(2-Diethylamino-ethyl)-3-hydroxy-3-(2-methox...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]ghrelin binding to human recombinant ghrelin receptor membrane preparationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed