Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50037557
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  1.51nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 308 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  4.60nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 308 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  4.10nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 303 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  2.30nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 288 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  3.30nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 273 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  2.60nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 293KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  3.20nMAssay Description:Dissociation constant for [3H]ORG2058 at human progesterone receptor at 298 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  2.70nMAssay Description:Dissociation constant for [3H]-ORG2058 at human progesterone receptor at 278 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  5.40nMAssay Description:Dissociation constant for [3H]-ORG2058 at human progesterone receptor at 310KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50422735(ORG-2058 | CHEMBL2311103)
Affinity DataKd:  2.5nMAssay Description:Dissociation constant for [3H]-ORG2058 at human progesterone receptor at 283 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.990nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 298 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.520nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 278 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataKd:  8.60nMAssay Description:Dissociation constant against Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  1.95nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 310KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.560nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 283 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.610nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 273 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  1.21nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 303 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM15336(1-methyl-3-(2-methylpropyl)-2,3,6,7-tetrahydro-1H-...)
Affinity DataKd:  5.90E+3nMAssay Description:Dissociation constant against Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.680nMAssay Description:Dissociation constant for [3H]R-1881 binding to human androgen receptor at 288 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM10849(CHEMBL113 | 1,3,7-trimethyl-3,7-dihydropurine-2,6-...)
Affinity DataKd:  4.50E+4nMAssay Description:Dissociation constant against Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM10847(Theophylline (1,3-dimethylxanthine) | 1,3-dimethyl...)
Affinity DataKd:  1.20E+4nMAssay Description:Dissociation constant against Adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataKd:  0.740nMAssay Description:Dissociation constant value of the radiolabeled compound against the androgen receptor 293 KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2012
Entry Details Article
PubMed