Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 1273
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10590({3-[(6-chloro-1,2,3,4-tetrahydroacridin-9-yl)amino...)
Affinity DataIC50: 0.290nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10586([3-({7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^...)
Affinity DataIC50: 0.320nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10585(7-chloro-15-methyl-N-[8-(1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 0.330nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10588(CHEMBL2011492 | 3-Chloro-6,7,10,11-tetrahydro-9-me...)
Affinity DataIC50: 0.330nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10584(7-chloro-15-methyl-N-[7-(1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 0.340nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10589(CHEMBL2011496 | 3-Chloro-6,7,10,11-tetrahydro-9-me...)
Affinity DataIC50: 0.400nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10587(7-chloro-N-{6-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 0.450nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10583(CHEMBL2011483 | 7-chloro-15-methyl-N-[6-(1,2,3,4-t...)
Affinity DataIC50: 0.5nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10592(7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^{2,11...)
Affinity DataIC50: 0.780nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10582(15-ethyl-N-[8-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 0.820nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10585(7-chloro-15-methyl-N-[8-(1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 4.74nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10582(15-ethyl-N-[8-(1,2,3,4-tetrahydroacridin-9-ylamino...)
Affinity DataIC50: 5.55nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10584(7-chloro-15-methyl-N-[7-(1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 6.70nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10588(CHEMBL2011492 | 3-Chloro-6,7,10,11-tetrahydro-9-me...)
Affinity DataIC50: 7.38nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10583(CHEMBL2011483 | 7-chloro-15-methyl-N-[6-(1,2,3,4-t...)
Affinity DataIC50: 7.69nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10589(CHEMBL2011496 | 3-Chloro-6,7,10,11-tetrahydro-9-me...)
Affinity DataIC50: 7.80nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10587(7-chloro-N-{6-[(6-chloro-1,2,3,4-tetrahydroacridin...)
Affinity DataIC50: 14nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10586([3-({7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^...)
Affinity DataIC50: 16.4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10590({3-[(6-chloro-1,2,3,4-tetrahydroacridin-9-yl)amino...)
Affinity DataIC50: 31.1nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 43.9nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 205nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10592(7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^{2,11...)
Affinity DataIC50: 236nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10441((+)-Huperzine A | (13E)-1-amino-13-ethylidene-11-m...)
Affinity DataIC50: 260nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed
TargetCholinesterase(Human)
Universitat De Barcelona

LigandPNGBDBM10441((+)-Huperzine A | (13E)-1-amino-13-ethylidene-11-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/8/2006
Entry Details Article
PubMed