Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50015931
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162568(6,7-Dichloro-2-cyclopentyl-5-[4-(2H-tetrazol-5-yl)...)
Affinity DataEC50:  122nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162580(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[5-(2H-tetra...)
Affinity DataEC50:  761nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162578(6,7-Dichloro-2,2-dimethyl-5-[4-(2H-tetrazol-5-yl)-...)
Affinity DataEC50:  782nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162579(2-Cyclopentyl-6,7-dimethyl-5-[3-(pyridin-4-ylsulfa...)
Affinity DataEC50:  596nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162574(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[3-(2H-tetra...)
Affinity DataEC50:  371nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162576(2-Butyl-6,7-dichloro-2-cyclopentyl-5-[4-(2H-tetraz...)
Affinity DataEC50:  1.09E+3nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162575(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[3-(pyridin-...)
Affinity DataEC50:  562nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162577(6,7-Dichloro-2-cyclopentyl-2-methyl-5-{2-[4-(2H-te...)
Affinity DataEC50:  276nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162572(6,7-Dichloro-2-cyclopentyl-5-[3-(pyridin-4-ylsulfa...)
Affinity DataEC50:  165nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162571(N-Acetyl-4-(6,7-dichloro-2-cyclopentyl-2-methyl-1-...)
Affinity DataEC50:  442nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162573(6,7-Dichloro-2-isopropyl-5-[4-(2H-tetrazol-5-yl)-b...)
Affinity DataEC50:  195nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162569(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[4-(2H-tetra...)
Affinity DataEC50:  223nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162570(2-(6,7-Dichloro-2-cyclopentyl-2-methyl-1-oxo-indan...)
Affinity DataEC50:  600nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162556(6,7-Dichloro-2-isopropyl-5-[3-(pyridin-4-ylsulfany...)
Affinity DataEC50:  839nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162566(6,7-Dichloro-2-propyl-5-[4-(2H-tetrazol-5-yl)-benz...)
Affinity DataEC50:  282nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162567(6,7-Dichloro-2-cyclopentyl-2-methyl-5-{2-[4-(2H-te...)
Affinity DataEC50:  1.16E+3nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162565(6,7-Dichloro-2-propyl-5-[3-(pyridin-4-ylsulfanylme...)
Affinity DataEC50:  186nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162564(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[4-(2H-tetra...)
Affinity DataEC50:  589nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162563(6,7-Dichloro-2-cyclopentyl-2-methyl-5-{3-[4-(2H-te...)
Affinity DataEC50:  270nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162562(6,7-Dichloro-2-methyl-2-phenyl-5-[4-(2H-tetrazol-5...)
Affinity DataEC50:  629nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162561(6,7-Dichloro-2-cyclopentyl-2-methyl-5-[3-(2H-tetra...)
Affinity DataEC50:  5.00E+3nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162560(N-[4-(6,7-Dichloro-2-cyclopentyl-2-methyl-1-oxo-in...)
Affinity DataEC50:  515nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162559(6,7-Dimethyl-2-propyl-5-[3-(pyridin-4-ylsulfanylme...)
Affinity DataEC50:  291nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162557(4-(6,7-Dichloro-2-cyclopentyl-2-methyl-1-oxo-indan...)
Affinity DataEC50:  892nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50162558(6,7-Dichloro-2-cyclopentyl-2-methyl-5-{4-[4-(2H-te...)
Affinity DataEC50:  225nMAssay Description:Binding affinity against metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed