Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50015876
TargetAlpha-1A adrenergic receptor(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50161871(Pyrazine-2-carboxylic acid {4-[4-(6-fluoro-benzo[b...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]prazosin binding to human adrenergic alpha-1A receptor expressed in CHO-K1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50161869(2-[(Z)-2,6-Dichloro-phenylimino]-6-{3-[4-(2-methox...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]prazosin binding to human adrenergic alpha-1A receptor expressed in CHO-K1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50161870(4-Amino-N-{2-[4-(1H-indol-4-yl)-piperidin-1-yl]-et...)
Affinity DataKi:  9.5nMAssay Description:Inhibition of [3H]prazosin binding to human adrenergic alpha-1A receptor expressed in CHO-K1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50161872(1-[2-(2,4-Dichloro-phenyl)-2-imidazol-1-ylmethyl-[...)
Affinity DataKi:  300nMAssay Description:Inhibition of [3H]prazosin binding to human adrenergic alpha-1A receptor expressed in CHO-K1 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed