Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50037545
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161753(N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-4-chlorobenza...)
Affinity DataIC50: 4.54E+3nMAssay Description:Functional antagonism of rat 5-hydroxytryptamine 3 receptor in cell-based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
LigandPNGBDBM50161753(N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-4-chlorobenza...)
Affinity DataKi:  27nMAssay Description:Inhibition of methyllycaconitine (MLA) binding to Nicotinic acetylcholine receptor alpha-7 in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50161753(N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-4-chlorobenza...)
Affinity DataKi:  1.66E+3nMAssay Description:Inhibition of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor from rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed