Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50015679
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataIC50: 0.261nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataIC50: 0.590nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159681((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...)
Affinity DataIC50: 0.623nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159684((S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 0.903nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159682((S)-1-[2-Amino-3-(4-hydroxy-2-methyl-phenyl)-propi...)
Affinity DataIC50: 0.924nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159681((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...)
Affinity DataIC50: 1.08nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataIC50: 2.31nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159686((S)-1-[2-Amino-3-(4-hydroxy-2-isopropyl-6-methyl-p...)
Affinity DataIC50: 10.6nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159682((S)-1-[2-Amino-3-(4-hydroxy-2-methyl-phenyl)-propi...)
Affinity DataIC50: 28.7nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataIC50: 46.4nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159684((S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 47.1nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159683((S)-1-[2-Amino-3-(4-hydroxy-2,6-diisopropyl-phenyl...)
Affinity DataIC50: 299nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159686((S)-1-[2-Amino-3-(4-hydroxy-2-isopropyl-6-methyl-p...)
Affinity DataIC50: 601nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159683((S)-1-[2-Amino-3-(4-hydroxy-2,6-diisopropyl-phenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159681((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...)
Affinity DataKi:  0.0630nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159684((S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-pr...)
Affinity DataKi:  0.0840nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataKi:  0.111nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159682((S)-1-[2-Amino-3-(4-hydroxy-2-methyl-phenyl)-propi...)
Affinity DataKi:  0.132nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159686((S)-1-[2-Amino-3-(4-hydroxy-2-isopropyl-6-methyl-p...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159683((S)-1-[2-Amino-3-(4-hydroxy-2,6-diisopropyl-phenyl...)
Affinity DataKi:  2.29nMAssay Description:Inhibition of [3H]DAMGO binding to mu-Opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataKi:  28.2nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159681((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...)
Affinity DataKi:  55.7nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159684((S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-pr...)
Affinity DataKi:  69.7nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159683((S)-1-[2-Amino-3-(4-hydroxy-2,6-diisopropyl-phenyl...)
Affinity DataKi:  105nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159686((S)-1-[2-Amino-3-(4-hydroxy-2-isopropyl-6-methyl-p...)
Affinity DataKi:  190nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159682((S)-1-[2-Amino-3-(4-hydroxy-2-methyl-phenyl)-propi...)
Affinity DataKi:  529nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159680((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...)
Affinity DataKi:  594nMAssay Description:Inhibition of [3H]DPDPE binding to delta-Opioid receptor More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed