Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 833
LigandPNGBDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM6071(thieno[3,2-b]pyridine-6-carbonitrile 14 | 7-[(2,4-...)
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6442(7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-{3-[(4-m...)
Affinity DataIC50: 21nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6441(thieno[3,2-b]pyridine-6-carbonitrile 13 | 7-[(2,4-...)
Affinity DataIC50: 34nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6084(thieno[3,2-b]pyridine-6-carbonitrile 37 | 7-[(2,4-...)
Affinity DataIC50: 50nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6439(7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-phenylth...)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6447(7-(2,4-dichlorophenoxy)-2-{4-[(4-methylpiperazin-1...)
Affinity DataIC50: 580nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6445(4-[(2,4-dichloro-5-methoxyphenyl)amino]-2-[4-(morp...)
Affinity DataIC50: 830nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6438(7-[(2,4-dichloro-5-methoxyphenyl)amino]thieno[3,2-...)
Affinity DataIC50: 2.50E+3nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6443(7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-{2-[(4-m...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed
LigandPNGBDBM6444(7-[(2,4-dichloro-5-methoxyphenyl)amino]-3-[4-(morp...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Kinase assays were performed using the europium/APC detection format (LANCE, Perkin Elmer). HTRF is based on the proximity of europium cryptate (dono...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2005
Entry Details Article
PubMed