Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 851
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
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LigandPNGBDBM6683({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 26nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
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LigandPNGBDBM6684({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 29nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50: 33nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
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LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 46nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
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LigandPNGBDBM6702(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 52nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50: 53nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6697(6-[(2,6-dichlorophenyl)carbonyl]-3-[(2,6-difluorop...)
Affinity DataIC50: 53nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50: 57nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50: 63nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50: 68nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50: 91nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50: 93nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 95nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50: 96nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50: 102nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50: 104nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6683({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 105nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50: 121nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50: 122nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50: 132nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6684({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 143nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 154nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50: 160nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6682({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 165nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50: 209nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6682({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 214nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50: 239nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50: 324nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50: 326nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 328nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50: 359nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6692(6-[(2-chlorophenyl)carbonyl]-3-[(2,6-difluoropheny...)
Affinity DataIC50: 428nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6684({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 464nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50: 475nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6699(6-[(2,6-difluorophenyl)carbonyl]-3-(thiophen-2-ylc...)
Affinity DataIC50: 547nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6695(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methoxyphen...)
Affinity DataIC50: 603nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6683({2-amino-6-[(2,6-difluorophenyl)carbonyl]imidazo[1...)
Affinity DataIC50: 786nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50: 810nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6704(6-[(2,6-dichlorophenyl)carbonyl]-3-({2,6-difluoro-...)
Affinity DataIC50: 812nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50: 827nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50: 838nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6705((2Z)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50: 896nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6703(6-[(2,6-dichlorophenyl)carbonyl]-3-({4-[2-(diethyl...)
Affinity DataIC50: 984nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50: 1.03E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6693(3-[(2,6-difluorophenyl)carbonyl]-6-{[2-(trifluorom...)
Affinity DataIC50: 1.07E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50: 1.08E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50: 1.14E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6694(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methylpheny...)
Affinity DataIC50: 1.29E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50: 1.55E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50: 1.69E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2005
Entry Details Article
PubMed
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