Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50015483
TargetDisintegrin and metalloproteinase domain-containing protein 9(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 9 (ADAM9)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 5.93nMAssay Description:Inhibition of A disintegrin and metalloprotease domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 7.5nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 17 (ADAM17, TACE)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 8.10nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 10 (ADAM10)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156477({3-(3-Bromo-phenyl)-2-[(furan-2-carbonyl)-amino]-a...)
Affinity DataIC50: 16.7nMAssay Description:Inhibition of A disintegrin and metalloprotease domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156475(2-[2-[(5-Bromo-furan-2-carbonyl)-amino]-3-(4-bromo...)
Affinity DataIC50: 24.8nMAssay Description:Inhibition of A disintegrin and metalloprotease domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156476(2-[2-Benzoylamino-3-(2-fluoro-phenyl)-acryloylamin...)
Affinity DataIC50: 40.5nMAssay Description:Inhibition of A disintegrin and metalloprotease domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156478(2-{2-[(Furan-2-carbonyl)-amino]-3-furan-2-yl-acryl...)
Affinity DataIC50: 42.3nMAssay Description:Inhibition of A disintegrin and metalloprotease domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156476(2-[2-Benzoylamino-3-(2-fluoro-phenyl)-acryloylamin...)
Affinity DataIC50: 1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 10 (ADAM10)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156477({3-(3-Bromo-phenyl)-2-[(furan-2-carbonyl)-amino]-a...)
Affinity DataIC50: 1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 10 (ADAM10)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Human)
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156478(2-{2-[(Furan-2-carbonyl)-amino]-3-furan-2-yl-acryl...)
Affinity DataIC50: 1.05E+4nMAssay Description:In vitro inhibition of A disintegrin and metalloprotease domain 10 (ADAM10)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed