Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50037467
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154301([(5S,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 40nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154297([(5S,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154295([(5S,9S,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154298([(5R,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154296([(5R,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154303([(5R,9R,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154308([(5R,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154299([(5S,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154305([(5R,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154304([(5S,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154302([(5S,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154300([(5S,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154309([(5R,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154306([(5R,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of [3H]DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM21015([tyrosyl-3,5-3H(N)]-D-Ala2-Mephe4-glyol5-enkephali...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154301([(5S,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154297([(5S,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154295([(5S,9S,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154298([(5R,9S,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154296([(5R,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154303([(5R,9R,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154308([(5R,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154306([(5R,9R,12R,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154305([(5R,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154299([(5S,9S,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  2.70E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154304([(5S,9R,12S,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154302([(5S,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154300([(5S,9S,12R,14aR)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50154309([(5R,9R,12S,14aS)-9-Benzyl-5-(4-hydroxy-benzyl)-12...)
Affinity DataKi:  2.30E+5nMAssay Description:Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed