Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50015299
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154167([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154170([1-(6-Chloro-1H-indazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154165([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154148([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154174([1-(1-Methyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 3.40nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154149([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154149([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154168([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 10nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154173([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154156([1-(1H-Pyrazol-3-ylaminooxalyl)-pentyl]-carbamic a...)
Affinity DataIC50: 18nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154155([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 20nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154171([1-(5-Phenyl-1H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 22nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154147([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154159([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 36nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154163([1-(2-Cyclobutyl-2H-pyrazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50: 45nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154160([1-(2-Cyclopropylmethyl-2H-pyrazol-3-ylaminooxalyl...)
Affinity DataIC50: 51nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154175([1-(2-Ethyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-ca...)
Affinity DataIC50: 52nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154172([1-(2-Isopropyl-2H-pyrazol-3-ylaminooxalyl)-pentyl...)
Affinity DataIC50: 54nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154146([1-(2-Cyclohexyl-2H-pyrazol-3-ylaminooxalyl)-penty...)
Affinity DataIC50: 58nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154169([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 62nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154176([1-(2-Phenyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 63nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154162([1-(2-Benzyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 65nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154164([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154157([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 68nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154151([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154150({1-[2-(3,3-Dimethyl-butyl)-2H-pyrazol-3-ylaminooxa...)
Affinity DataIC50: 71nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154153([1-(2-Isobutyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]...)
Affinity DataIC50: 76nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154152([1-(2-Cyclopentyl-2H-pyrazol-3-ylaminooxalyl)-pent...)
Affinity DataIC50: 83nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154166([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 120nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154158([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 135nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154145([1-(1-Phenyl-ethylaminooxalyl)-pentyl]-carbamic ac...)
Affinity DataIC50: 140nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154154([1-(Isoxazol-3-ylaminooxalyl)-pentyl]-carbamic aci...)
Affinity DataIC50: 350nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50154161([1-(2-Methyl-2H-pyrazol-3-ylaminooxalyl)-pentyl]-c...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory potency against human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed