Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 50015246
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153406(Trifluoro-acetate3-{(R)-4-[4-((S)-1-carboxy-2-meth...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153384(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153395(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153412(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153398(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153415(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153396(Trifluoro-acetate3-{(S)-2-[4-((S)-1-carboxy-2-meth...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153403(Trifluoro-acetate3-{(S)-2-[4-(1-carboxy-2-methyl-p...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153418(Trifluoro-acetate3-{(S)-2-[4-(1-carboxy-pentyloxy)...)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153409(Trifluoro-acetate3-{(S)-2-[4-(1-carboxy-propoxy)-b...)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153413(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153411(Trifluoro-acetate3-{(S)-2-[4-(1-carboxy-butoxy)-be...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153402(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153400(Trifluoro-acetate3-{(S)-2-[4-((S)-1-carboxy-ethoxy...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153405(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153388(Trifluoro-acetate1-benzyl-3-{(S)-2-[4-((R)-1-carbo...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153419(Trifluoro-acetate3-{(S)-2-[4-(1-carboxy-ethoxy)-be...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153417(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153389(Trifluoro-acetate3-[(R)-4-(4-carboxymethyl-benzylc...)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153401(Trifluoro-acetate1-(2-fluoro-benzyl)-3-oxo-3-{(S)-...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153385(Trifluoro-acetate3-[(S)-2-(4-carboxy-benzylcarbamo...)
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153387(Trifluoro-acetate3-[(S)-2-(4-carboxy-benzylcarbamo...)
Affinity DataIC50: 75nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153391(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-ethoxy...)
Affinity DataIC50: 82nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153381(Trifluoro-acetate1-(2-fluoro-benzyl)-3-[(R)-4-(4-m...)
Affinity DataIC50: 87nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153408(Trifluoro-acetate3-[(S)-2-(4-carboxymethoxy-benzyl...)
Affinity DataIC50: 118nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153399(Trifluoro-acetate1-benzyl-3-[(R)-4-(4-carboxymethy...)
Affinity DataIC50: 161nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153394(Trifluoro-acetate1-(2-fluoro-benzyl)-3-[(S)-2-(4-m...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153393(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 295nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153404(Trifluoro-acetate2-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 450nMAssay Description:Inhibition of Dipeptidylpeptidase IXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153410(Trifluoro-acetate1-benzyl-3-[(S)-2-(4-carboxy-benz...)
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153407(Trifluoro-acetate3-((S)-2-benzylcarbamoyl-pyrrolid...)
Affinity DataIC50: 539nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153386(Trifluoro-acetate1-(2-fluoro-benzyl)-3-oxo-3-[(S)-...)
Affinity DataIC50: 721nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50153386(Trifluoro-acetate1-(2-fluoro-benzyl)-3-oxo-3-[(S)-...)
Affinity DataIC50: 870nMAssay Description:Inhibition of human Potassium channel HERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153397(Trifluoro-acetate1-benzyl-3-[(S)-2-(2-carboxy-benz...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153416(Trifluoro-acetate1-benzyl-3-[(S)-2-(3-carboxy-benz...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153390(Trifluoro-acetate1-(2-fluoro-benzyl)-3-{(S)-2-[4-(...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153383((S)-1-(3-Amino-4-phenyl-butyryl)-pyrrolidine-2-car...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153392(Trifluoro-acetate2-[(S)-2-(3-carboxy-benzylcarbamo...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153380(Trifluoro-acetate2-[(S)-2-(2-carboxy-benzylcarbamo...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153404(Trifluoro-acetate2-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of Dipeptidylpeptidase VIIIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153414(Trifluoro-acetate2-[(S)-2-(4-carboxy-benzylcarbamo...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153386(Trifluoro-acetate1-(2-fluoro-benzyl)-3-oxo-3-[(S)-...)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Dipeptidylpeptidase VIIIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153404(Trifluoro-acetate2-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human recombinant Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50153381(Trifluoro-acetate1-(2-fluoro-benzyl)-3-[(R)-4-(4-m...)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of human Potassium channel HERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153384(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of Fibroblast activation protein alpha (seprase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153384(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of prolyl endopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProlyl endopeptidase FAP(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153382(Trifluoro-acetate3-{(S)-2-[4-((R)-1-carboxy-2-meth...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of Fibroblast activation protein alpha (seprase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153389(Trifluoro-acetate3-[(R)-4-(4-carboxymethyl-benzylc...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Dipeptidylpeptidase VIIIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50153386(Trifluoro-acetate1-(2-fluoro-benzyl)-3-oxo-3-[(S)-...)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of Quiescent cell prolyl dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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