Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50036011
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005120(Nemonapride | N-((2S,3S)-1-Benzyl-2-methyl-pyrroli...)
Affinity DataIC50: 0.490nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataIC50: 17nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataIC50: 32nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM81774(Sulpiride-S | CAS_15676-16-1 | Sulpiride-l | SULPI...)
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM81774(Sulpiride-S | CAS_15676-16-1 | Sulpiride-l | SULPI...)
Affinity DataIC50: 233nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM48320(SMR000058471 | METOCLOPRAMIDE | METOCLOPRAMIDE HYD...)
Affinity DataIC50: 820nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005121(CHEMBL308129 | (R)3,5-Dichloro-N-(1-ethyl-pyrrolid...)
Affinity DataIC50: 2.92E+3nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005120(Nemonapride | N-((2S,3S)-1-Benzyl-2-methyl-pyrroli...)
Affinity DataKi:  0.120nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  2.20nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  9.5nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM50005117((racemic)5'-(5-Ethanesulfonyl-2-methoxy-phenyl)-1-...)
Affinity DataKi:  29nMAssay Description:Compound was evaluated for binding affinity towards Dopamine receptor D2 using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM81774(Sulpiride-S | CAS_15676-16-1 | Sulpiride-l | SULPI...)
Affinity DataKi:  39nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM48320(SMR000058471 | METOCLOPRAMIDE | METOCLOPRAMIDE HYD...)
Affinity DataKi:  104nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Lund

Curated by ChEMBL
LigandPNGBDBM48320(SMR000058471 | METOCLOPRAMIDE | METOCLOPRAMIDE HYD...)
Affinity DataKi:  104nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed