Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50015130
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151832(2-{(R)-4-[3-Amino-4-((R)-2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151840((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2,4...)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151828(2-{(R)-4-[(R)-3-Amino-4-(3,4-difluoro-phenyl)-buty...)
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151836(2-{4-[(R)-3-Amino-4-(2-fluoro-phenyl)-butyryl]-3-b...)
Affinity DataIC50: 34nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151842(2-{4-[3-Amino-4-((R)-3,4-difluoro-phenyl)-butyryl]...)
Affinity DataIC50: 44nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151844((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2,5...)
Affinity DataIC50: 51nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151829((R)-3-Amino-1-((R)-3-benzyl-morpholin-4-yl)-4-(2-f...)
Affinity DataIC50: 108nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151835(2-{(R)-4-[(R)-3-Amino-4-(2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 114nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151825(2-[4-((R)-3-Amino-4-phenyl-butyryl)-3-benzyl-piper...)
Affinity DataIC50: 134nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151843((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2-f...)
Affinity DataIC50: 139nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151833((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-thiazol-4...)
Affinity DataIC50: 143nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151820((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-pyridin-3...)
Affinity DataIC50: 155nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151834((R)-3-Amino-1-[(R)-2-(4-fluoro-benzyl)-piperazin-1...)
Affinity DataIC50: 166nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151838((R)-3-Amino-1-((R)-2-benzyl-4-methyl-piperazin-1-y...)
Affinity DataIC50: 225nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151822(2-{(S)-4-[(R)-3-Amino-4-(3,4-difluoro-phenyl)-buty...)
Affinity DataIC50: 280nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151839((R)-3-Amino-1-((R)-2,4-dibenzyl-piperazin-1-yl)-4-...)
Affinity DataIC50: 405nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151842(2-{4-[3-Amino-4-((R)-3,4-difluoro-phenyl)-butyryl]...)
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151831((R)-3-Amino-4-(2-fluoro-phenyl)-1-[(R)-2-(4-fluoro...)
Affinity DataIC50: 610nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151828(2-{(R)-4-[(R)-3-Amino-4-(3,4-difluoro-phenyl)-buty...)
Affinity DataIC50: 640nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151827(2-{(S)-4-[3-Amino-4-((R)-2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 690nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151826((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-isopropyl...)
Affinity DataIC50: 922nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151841((R)-3-Amino-1-((S)-2-benzyl-piperidin-1-yl)-4-(2-f...)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151822(2-{(S)-4-[(R)-3-Amino-4-(3,4-difluoro-phenyl)-buty...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151824((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-methyl-pi...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151805(CHEMBL184262 (24) | CHEMBL184262 | (R)-3-Amino-4-p...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151819((R)-3-Amino-4-(2-fluoro-phenyl)-1-piperazin-1-yl-b...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151825(2-[4-((R)-3-Amino-4-phenyl-butyryl)-3-benzyl-piper...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151823(2-[4-((S)-2-Amino-3-phenyl-propyl)-3-benzyl-pipera...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151827(2-{(S)-4-[3-Amino-4-((R)-2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151836(2-{4-[(R)-3-Amino-4-(2-fluoro-phenyl)-butyryl]-3-b...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151839((R)-3-Amino-1-((R)-2,4-dibenzyl-piperazin-1-yl)-4-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151830(2-{4-[(S)-3-Amino-4-(3,4-difluoro-phenyl)-butyryl]...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151837(2-{4-[3-Amino-4-((S)-2-fluoro-phenyl)-butyryl]-3-b...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151821(2-[4-((S)-3-Amino-4-phenyl-butyryl)-3-benzyl-piper...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151832(2-{(R)-4-[3-Amino-4-((R)-2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151831((R)-3-Amino-4-(2-fluoro-phenyl)-1-[(R)-2-(4-fluoro...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151837(2-{4-[3-Amino-4-((S)-2-fluoro-phenyl)-butyryl]-3-b...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151821(2-[4-((S)-3-Amino-4-phenyl-butyryl)-3-benzyl-piper...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151830(2-{4-[(S)-3-Amino-4-(3,4-difluoro-phenyl)-butyryl]...)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibitory concentration against Dipeptidylpeptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151826((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-isopropyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151844((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2,5...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151835(2-{(R)-4-[(R)-3-Amino-4-(2-fluoro-phenyl)-butyryl]...)
Affinity DataIC50: 6.60E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151840((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2,4...)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151841((R)-3-Amino-1-((S)-2-benzyl-piperidin-1-yl)-4-(2-f...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151819((R)-3-Amino-4-(2-fluoro-phenyl)-1-piperazin-1-yl-b...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151843((R)-3-Amino-1-((R)-2-benzyl-piperazin-1-yl)-4-(2-f...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151833((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-thiazol-4...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151838((R)-3-Amino-1-((R)-2-benzyl-4-methyl-piperazin-1-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151820((R)-3-Amino-4-(2-fluoro-phenyl)-1-((R)-2-pyridin-3...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151834((R)-3-Amino-1-[(R)-2-(4-fluoro-benzyl)-piperazin-1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline peptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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