Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50015129
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151798([6-(2,4-Dichloro-phenyl)-2-(3,5-dimethoxy-phenyl)-...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM15564(CHEMBL363319 | (3R)-3-amino-1-(1,3-thiazolidin-3-y...)
Affinity DataIC50: 119nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151804((R)-3-Amino-4-(2,5-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 270nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151793((R)-3-Amino-4-(2,4-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 589nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151803((R)-3-Amino-4-(2-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 931nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151789((R)-3-Amino-1-thiazolidin-3-yl-4-o-tolyl-butan-1-o...)
Affinity DataIC50: 981nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151796((R)-3-Amino-4-(4-nitro-phenyl)-1-thiazolidin-3-yl-...)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151794((R)-3-Amino-4-(3,4-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM11557((2S)-1-[(3R)-3-amino-4-phenylbutanoyl]-N-({5-chlor...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151817((R)-3-Amino-4-(3-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151799((R)-3-Amino-4-(3,4-dichloro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151810((R)-3-Amino-1-thiazolidin-3-yl-4-(2-trifluoromethy...)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151800(2-((R)-2-Amino-4-oxo-4-thiazolidin-3-yl-butyl)-ben...)
Affinity DataIC50: 2.52E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151805(CHEMBL184262 (24) | CHEMBL184262 | (R)-3-Amino-4-p...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151807((R)-3-Amino-4-(4-chloro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151791((R)-3-Amino-4-(4-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151816((R)-3-Amino-1-thiazolidin-3-yl-4-(3-trifluoromethy...)
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151808((R)-3-Amino-1-thiazolidin-3-yl-4-thiophen-3-yl-but...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151809((R)-3-Amino-4-(4-iodo-phenyl)-1-thiazolidin-3-yl-b...)
Affinity DataIC50: 5.78E+3nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151806((R)-3-Amino-1-thiazolidin-3-yl-4-(4-trifluoromethy...)
Affinity DataIC50: 7.69E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151812((R)-3-Amino-4-(2,6-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 8.48E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151792(3-((R)-2-Amino-4-oxo-4-thiazolidin-3-yl-butyl)-ben...)
Affinity DataIC50: 8.95E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151797((R)-3-Amino-4-(2,3-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151809((R)-3-Amino-4-(4-iodo-phenyl)-1-thiazolidin-3-yl-b...)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151813(4-((R)-2-Amino-4-oxo-4-thiazolidin-3-yl-butyl)-ben...)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151811((R)-3-Amino-5-phenyl-1-thiazolidin-3-yl-pentan-1-o...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151796((R)-3-Amino-4-(4-nitro-phenyl)-1-thiazolidin-3-yl-...)
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151816((R)-3-Amino-1-thiazolidin-3-yl-4-(3-trifluoromethy...)
Affinity DataIC50: 2.46E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM15564(CHEMBL363319 | (3R)-3-amino-1-(1,3-thiazolidin-3-y...)
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151795((R)-3-Amino-4-cyclopentyl-1-thiazolidin-3-yl-butan...)
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151792(3-((R)-2-Amino-4-oxo-4-thiazolidin-3-yl-butyl)-ben...)
Affinity DataIC50: 2.98E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151814((R)-3-Amino-4-cyclohexyl-1-thiazolidin-3-yl-butan-...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151794((R)-3-Amino-4-(3,4-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151807((R)-3-Amino-4-(4-chloro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151802((R)-3-Amino-4-pyridin-2-yl-1-thiazolidin-3-yl-buta...)
Affinity DataIC50: 3.96E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151815((R)-3-Amino-4-pyridin-3-yl-1-thiazolidin-3-yl-buta...)
Affinity DataIC50: 4.49E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151790((R)-3-Amino-4-furan-3-yl-1-thiazolidin-3-yl-butan-...)
Affinity DataIC50: 4.69E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151799((R)-3-Amino-4-(3,4-dichloro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 4.85E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151817((R)-3-Amino-4-(3-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 4.85E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151803((R)-3-Amino-4-(2-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 4.97E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151801((R)-3-Amino-4-pyridin-4-yl-1-thiazolidin-3-yl-buta...)
Affinity DataIC50: 5.10E+4nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151793((R)-3-Amino-4-(2,4-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 5.61E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151791((R)-3-Amino-4-(4-fluoro-phenyl)-1-thiazolidin-3-yl...)
Affinity DataIC50: 6.76E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151804((R)-3-Amino-4-(2,5-difluoro-phenyl)-1-thiazolidin-...)
Affinity DataIC50: 7.76E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151810((R)-3-Amino-1-thiazolidin-3-yl-4-(2-trifluoromethy...)
Affinity DataIC50: 8.21E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151789((R)-3-Amino-1-thiazolidin-3-yl-4-o-tolyl-butan-1-o...)
Affinity DataIC50: 9.21E+4nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151805(CHEMBL184262 (24) | CHEMBL184262 | (R)-3-Amino-4-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 2(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151800(2-((R)-2-Amino-4-oxo-4-thiazolidin-3-yl-butyl)-ben...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against quiescent cell proline dipeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50151818((S)-3-Amino-3-phenyl-1-thiazolidin-3-yl-propan-1-o...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against Dipeptidyl peptidase IVMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed