Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50000369
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004801(CHEMBL137648 | 3-(3-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004808(CHEMBL134400 | 3-Benzyl-8-[4-(4-fluoro-phenyl)-4-o...)
Affinity DataKi:  0.0230nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004819(CHEMBL135917 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0290nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004817(CHEMBL135832 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0330nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004803(CHEMBL337149 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0350nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004805(CHEMBL136852 | 3-Butyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.0360nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004807(CHEMBL334349 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0390nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004816(CHEMBL137309 | 3-(2-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004810(CHEMBL135722 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0470nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004818(CHEMBL136942 | 3-Ethyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.0570nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.0580nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004802(CHEMBL135316 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0620nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004804(CHEMBL135500 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0630nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004815(CHEMBL344399 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0630nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004806(CHEMBL134545 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0670nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004800(CHEMBL538404 | 3-(4-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  0.0690nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004812(CHEMBL335606 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0870nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004819(CHEMBL135917 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0960nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004813(8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-methyl-1-phe...)
Affinity DataKi:  0.118nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004809(CHEMBL337181 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.119nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004814(CHEMBL135860 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004807(CHEMBL334349 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.130nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004811(CHEMBL335714 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.213nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004818(CHEMBL136942 | 3-Ethyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004805(CHEMBL136852 | 3-Butyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.410nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.450nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004813(8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]-3-methyl-1-phe...)
Affinity DataKi:  0.550nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004814(CHEMBL135860 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.680nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004803(CHEMBL337149 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  1nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004802(CHEMBL135316 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  1.10nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004815(CHEMBL344399 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  1.30nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004810(CHEMBL135722 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  1.90nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004808(CHEMBL134400 | 3-Benzyl-8-[4-(4-fluoro-phenyl)-4-o...)
Affinity DataKi:  3.20nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004816(CHEMBL137309 | 3-(2-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  4.40nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004801(CHEMBL137648 | 3-(3-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  5.30nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004817(CHEMBL135832 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  9.60nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004812(CHEMBL335606 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  12nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004809(CHEMBL337181 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  14nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004804(CHEMBL135500 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  19nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004800(CHEMBL538404 | 3-(4-Fluoro-benzyl)-8-[4-(4-fluoro-...)
Affinity DataKi:  21nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004806(CHEMBL134545 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  37nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50004811(CHEMBL335714 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  89nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed