Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50036041
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against HIV-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 185nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibitory concentration against HIV-2 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 275nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:In vitro Inhibitory activity against HIV-2 protease in the presence of 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:In vitro Inhibitory activity against HIV-2 protease in the presence of 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibitory concentration against HIV-2 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 725nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 975nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro Inhibitory activity against HIV-2 protease in the presence of 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory concentration against reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory concentration against pepsinMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against cathepsin DMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIV-2 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory concentration against HIV-1 protease in the absence of DMSOMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
