Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50015024
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150431(N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phen...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150430(N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phen...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150439(N*2*-Phenethyl-N*4*-((S)-1-phenyl-ethyl)-pyridine-...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150428(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-((S)-1-phen...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150425(N*4*-(2-Phenoxy-ethyl)-N*2*-((S)-1-phenyl-ethyl)-p...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150446(N*2*-(2-Phenoxy-ethyl)-N*4*-((S)-1-phenyl-ethyl)-p...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150441(N*2*-[2-(4-Fluoro-phenyl)-ethyl]-N*4*-((S)-1-pheny...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150422(N*2*-Phenethyl-N*4*-((S)-1-phenyl-ethyl)-pyrimidin...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150438(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-(1-phenyl-e...)
Affinity DataKi:  1nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150433(N*2*-(2-Phenoxy-ethyl)-N*4*-((S)-1-phenyl-ethyl)-p...)
Affinity DataKi:  2nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150436(N*4*-Phenethyl-N*2*-((S)-1-phenyl-ethyl)-pyridine-...)
Affinity DataKi:  3nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150437(N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-e...)
Affinity DataKi:  4nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150432(N*4*-[2-(4-Fluoro-phenyl)-ethyl]-N*2*-((S)-1-pheny...)
Affinity DataKi:  4nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150440(N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-pyrid...)
Affinity DataKi:  4nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150423(N-[2-(4-Fluoro-phenyl)-ethyl]-N''-((S)-1-phenyl-et...)
Affinity DataKi:  5nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150424(N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-e...)
Affinity DataKi:  5nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150442(N*4*-Phenethyl-N*2*-(1-phenyl-ethyl)-pyrimidine-2,...)
Affinity DataKi:  6nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150444(N*2*-[2-(4-Fluoro-phenyl)-ethyl]-N*4*-(1-phenyl-et...)
Affinity DataKi:  6nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150428(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-((S)-1-phen...)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150427(N-Phenethyl-N''-((S)-1-phenyl-ethyl)-pyridine-3,5-...)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150431(N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phen...)
Affinity DataKi:  15nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150426(N-[2-(4-Fluoro-phenyl)-ethyl]-N''-((S)-1-phenyl-et...)
Affinity DataKi:  16nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150445(N-Phenethyl-N''-((S)-1-phenyl-ethyl)-pyrimidine-4,...)
Affinity DataKi:  33nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150438(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-(1-phenyl-e...)
Affinity DataKi:  40nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150431(N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phen...)
Affinity DataKi:  370nMAssay Description:Binding affinity against D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150437(N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-e...)
Affinity DataKi:  476nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150429(N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-benze...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150438(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-(1-phenyl-e...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150428(N*4*-[2-(4-Fluoro-phenoxy)-ethyl]-N*2*-((S)-1-phen...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150437(N-[2-(4-Fluoro-phenoxy)-ethyl]-N''-((S)-1-phenyl-e...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150430(N*2*-[2-(4-Fluoro-phenoxy)-ethyl]-N*4*-((S)-1-phen...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150443(N-Phenethyl-N''-((S)-1-phenyl-ethyl)-benzene-1,3-d...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150435(N-(2-Phenoxy-ethyl)-N''-((S)-1-phenyl-ethyl)-pyrid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50150434(N-Phenethyl-N''-((S)-1-phenyl-ethyl)-pyridine-2,6-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against 5-Hydroxy tryptamine 7 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed