Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50014934
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50074242(CHEMBL23794 | (2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Acety...)
Affinity DataKd:  100nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50149285(3-{5-[3-(4-Fluoro-phenyl)-2-imino-4-oxo-thiazolidi...)
Affinity DataKd:  1.20E+4nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50149286(3-{5-[2,4-Dioxo-3-(p-tolylcarbamoyl-methyl)-thiazo...)
Affinity DataKd:  6.00E+3nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50149287(2-[(E)-2-(3-Bromo-2-hydroxy-5-nitro-phenyl)-vinyl]...)
Affinity DataKd:  6.00E+3nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50074243((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataKd:  1.50E+3nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50074251((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataKd:  2.70E+4nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50077198((S)-4-(4-Methoxy-benzylcarbamoyl)-4-{(S)-2-(2-naph...)
Affinity DataKd:  3.00E+3nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50149288(5-(2-Methoxy-5-nitro-benzylsulfanyl)-[1,3,4]thiadi...)
Affinity DataKd:  4.00E+3nMAssay Description:Dissociation constant for p56 Lck tyrosine kinase SH2 domain binding to C-terminal ITAM2 phosphopeptideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed