Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50014933
TargetPlasminogen activator inhibitor 1(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149275([{1-benzyl-5-[4-(trifluoromethoxy)phenyl]-1H-indol...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity of compound towards latent Plasminogen activator inhibitor-1 expressed as apparent KdMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149275([{1-benzyl-5-[4-(trifluoromethoxy)phenyl]-1H-indol...)
Affinity DataKd:  480nMAssay Description:Binding affinity to towards NBD-labeled S119C Plasminogen activator inhibitor-1 mutant in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149275([{1-benzyl-5-[4-(trifluoromethoxy)phenyl]-1H-indol...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50104518(CHEMBL544314 | CHEMBL40180 | 3-[1-[5-(2-Dimethylam...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149272([1-(4-tert-Butyl-benzyl)-5-m-tolyl-1H-indol-3-yl]-...)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149273([1-Benzyl-5-(3-trifluoromethoxy-phenyl)-1H-indol-3...)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149281([1-(4-tert-Butyl-benzyl)-5-(3-tert-butyl-phenyl)-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149282([1-Benzyl-7-(4-trifluoromethoxy-phenyl)-1H-indol-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149284(2-Hydroxy-4-(2-phenyl-4,5-dihydro-benzo[e]indol-3-...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149274(2-[4-(3,4-Dichloro-phenylcarbamoyl)-benzylamino]-4...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149276([1-(4-tert-Butyl-benzyl)-5-(4-trifluoromethoxy-phe...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149278([1-Benzyl-6-(4-trifluoromethoxy-phenyl)-1H-indol-3...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149277([1-(4-tert-Butyl-benzyl)-5-(3-methoxy-phenyl)-1H-i...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149283((1-Benzyl-6-phenyl-1H-indol-3-yl)-oxo-acetic acid ...)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149271([1-(4-Fluoro-benzyl)-6-phenyl-1H-indol-3-yl]-oxo-a...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149280([1-(4-tert-Butyl-benzyl)-6-(4-trifluoromethoxy-phe...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen activator inhibitor 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149279([1-Benzyl-4-(4-trifluoromethoxy-phenyl)-1H-indol-3...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human plasminogen activator inhibitor-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed