Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50014926
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149195(1-Benzyl-2,3-dihydro-1H-indole-5-carboxylic acid [...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223715(CHEMBL3706732)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223717(CHEMBL3706727)
Affinity DataIC50: 82nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149199(6-Hydroxy-2,5,7,8-tetramethyl-chroman-2-carboxylic...)
Affinity DataIC50: 147nMAssay Description:Inhibitory activity against on human calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223716(CHEMBL3706728)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibitory activity against on calpain 1 in C6 glial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50223715(CHEMBL3706732)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibitory activity against on calpain in C6 glial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Human)
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50149195(1-Benzyl-2,3-dihydro-1H-indole-5-carboxylic acid [...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against on calpain in C6 glial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed