Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50014872
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148588(ethyl hydrogen heptylphosphonate | Heptyl-phosphon...)
Affinity DataIC50: 1.06E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148590(Heptyl-phosphonic acid 1,3-dioxo-1,3-dihydro-isoin...)
Affinity DataIC50: 1.31E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148587(Heptyl-phosphonic acid mono-[2-(1,3-dioxo-1,3-dihy...)
Affinity DataIC50: 1.47E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148586(Butyl-phosphonic acid ethyl ester 3-phenoxy-benzyl...)
Affinity DataIC50: 2.01E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148593(N-HEXYLPHOSPHONATE ETHYL ESTER | ethyl hydrogen he...)
Affinity DataIC50: 3.56E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148585(Hexyl-phosphonic acid mono-[2-(1,3-dioxo-1,3-dihyd...)
Affinity DataIC50: 4.39E+3nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148594((1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-methyl et...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148583(Nonyl-phosphonic acid ethyl ester 3-phenoxy-benzyl...)
Affinity DataIC50: 1.48E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148596(Heptyl-phosphonic acid ethyl ester 3-phenoxy-benzy...)
Affinity DataIC50: 2.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148582(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethylet...)
Affinity DataIC50: 2.57E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148597(Tetradecyl-phosphonic acid 1,3-dioxo-1,3-dihydro-i...)
Affinity DataIC50: 4.10E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148584(Hexyl-phosphonic acid ethyl ester 3-phenoxy-benzyl...)
Affinity DataIC50: 4.26E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148591(2-(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)-ethyl e...)
Affinity DataIC50: 5.07E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148592(Nonyl-phosphonic acid 1,3-dioxo-1,3-dihydro-isoind...)
Affinity DataIC50: 8.71E+4nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148589(Butyl-phosphonic acid monoethyl ester | ethyl hydr...)
Affinity DataIC50: 4.31E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148595(Nonyl-phosphonic acid monoethyl ester | ethyl hydr...)
Affinity DataIC50: 4.71E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDiacylglycerol acyltransferase/mycolyltransferase Ag85C(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50148581(Tetradecyl-phosphonic acid ethyl ester 3-phenoxy-b...)
Affinity DataIC50: 8.62E+5nMAssay Description:In vitro concentration required to inhibit antigen 85C mycolyltransferase activity in Mycobacterium tuberculosisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed