Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50014857
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148365(2-{3-[4-(3,5-Bis-trifluoromethyl-benzyloxy)-phenyl...)
Affinity DataIC50: 390nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148366(2-{3-[4-(3-Chloro-benzyloxy)-phenyl]-1-phenyl-prop...)
Affinity DataIC50: 680nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50085942(2-{3-[3-(3,5-Dichloro-phenoxy)-phenyl]-hept-2-enyl...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148358(2-{(E)-3-[3,5-Bis-(4-chloro-benzyloxy)-phenyl]-all...)
Affinity DataIC50: 2.10E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148359(2-[3-(3-m-Tolyloxy-phenyl)-heptyl]-[1,2,4]oxadiazo...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148360(2-{(E)-3-[3-(Biphenyl-2-ylmethoxy)-phenyl]-but-2-e...)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148367(2-{(E)-3-[3,5-Bis-(4-trifluoromethyl-benzyloxy)-ph...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148368(2-{(E)-3-[4-(3,4-Dichloro-benzyloxy)-3-methoxy-phe...)
Affinity DataIC50: 3.22E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148363(2-{(E)-3-[2-Chloro-5-(3,4-dichloro-benzyloxy)-phen...)
Affinity DataIC50: 3.80E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50085963(2-{3-[3-(3,5-Bis-trifluoromethyl-phenoxymethyl)-ph...)
Affinity DataIC50: 5.29E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148364(2-{(E)-1-Methyl-3-[4-(3-trifluoromethyl-benzyloxy)...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148361(2-{(E)-3-[4-(3,4-Dichloro-benzyloxy)-phenyl]-1-met...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148362(2-{(Z)-3-[3-(3,5-Bis-trifluoromethyl-phenoxymethyl...)
Affinity DataIC50: 7.20E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148357(2-{(E)-3-[4-(3,5-Bis-trifluoromethyl-benzyloxy)-ph...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50085960(2-{(E)-3-[3-(3,5-Bis-trifluoromethyl-benzyloxy)-ph...)
Affinity DataIC50: 9.40E+3nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50148356(2-{(E)-3-[4-(3,5-Bis-trifluoromethyl-benzyloxy)-ph...)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibitory activity against tissue type plasminogen activatorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTissue-type plasminogen activator(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50085953(2-{3-[3-(Pyridin-2-ylmethoxy)-phenyl]-but-2-enyl}-...)
Affinity DataIC50: 2.40E+4nMAssay Description:In vitro concentration required for inhibition of tissue type plasminogen activator by plasminogen activator inhibitor-1 at concentration 25 umMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed