Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50035389
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50366912(CHEMBL1790774)
Affinity DataIC50: 0.590nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50366909(CHEMBL1790773)
Affinity DataIC50: 1.5nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50366908(CHEMBL1790772)
Affinity DataIC50: 9.60nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50146530((S)-2-[4-(4-{(S)-1-[(S)-1-((S)-2-Butylcarbamoyl-1-...)
Affinity DataIC50: 123nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50366910(CHEMBL1790776)
Affinity DataIC50: 135nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50366911(CHEMBL1790775)
Affinity DataIC50: 396nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50146528(6-Amino-2-(S)-amino-hexanoic acid [4-(6-methoxy-qu...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro concentration required for inhibition of Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50146524((S)-3-(S)-Hydroxy-4-{(S)-3-methyl-2-[2-(naphthalen...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed
TargetPlasmepsin II(Plasmodium falciparum)
University of Milan

Curated by ChEMBL
LigandPNGBDBM50223627(CHEMBL3215350)
Affinity DataKi:  180nMAssay Description:In vitro binding affinity towards Plasmodium falciparum plasmepsin-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/10/2012
Entry Details Article
PubMed