Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50014680
Target5-hydroxytryptamine receptor 1A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146087(1,3-Dimethyl-8-[4-(4-phenyl-piperazin-1-yl)-butyl]...)
Affinity DataKi:  2.10nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 1A receptor in vitro in hippocampus of the rat brain using [3H]8-OH-DPAT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146094(8-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi:  10.4nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 1A receptor in vitro in hippocampus of the rat brain using [3H]8-OH-DPAT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146089(1,3-dimethyl-9-{3-[4-(2'-methoxyphenyl)-piperazin-...)
Affinity DataKi:  17.2nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 1A receptor in vitro in hippocampus of the rat brain using [3H]8-OH-DPAT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146084(1,3-Dimethyl-8-[3-(4-phenyl-piperazin-1-yl)-propyl...)
Affinity DataKi:  25nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 1A receptor in vitro in hippocampus of the rat brain using [3H]8-OH-DPAT radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146087(1,3-Dimethyl-8-[4-(4-phenyl-piperazin-1-yl)-butyl]...)
Affinity DataKi:  243nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 2A receptor in vitro in cortex of the rat brain using [3H]ketanserin radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146089(1,3-dimethyl-9-{3-[4-(2'-methoxyphenyl)-piperazin-...)
Affinity DataKi:  562nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 2A receptor in vitro in cortex of the rat brain using [3H]ketanserin radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146094(8-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyl}...)
Affinity DataKi:  3.88E+3nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 2A receptor in vitro in cortex of the rat brain using [3H]ketanserin radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Collegium Medicum of The Jagiellonian University

Curated by ChEMBL
LigandPNGBDBM50146084(1,3-Dimethyl-8-[3-(4-phenyl-piperazin-1-yl)-propyl...)
Affinity DataKi:  4.68E+3nMAssay Description:Ability to bind to central serotonin 5-hydroxytryptamine 2A receptor in vitro in cortex of the rat brain using [3H]ketanserin radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed